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Search results for 'ilo'
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Starting at: $800.00
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Imiloxan hydrochloride
Imiloxan hydrochloride is a moderately potent, but highly selective α2-adrenoceptor antagonist, the only reported selective antagonist at the α2B-adrenoceptor not having potent α1-adrenoceptor antagonist activity. Learn MoreStarting at: $90.00
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Iloprost
Iloprost is a prostacyclin (PGI2) analog that inhibits platelet aggregation induced by collagen, thrombin and ADP with IC50 values of 0.24, 0.71 and 1.07 nM respectively. Learn MoreStarting at: $239.00
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Pilocarpine hydrochloride
Pilocarpine hydrochloride is a muscarinic agonist. Learn MoreStarting at: $49.00
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Psilocin
PsilocinNon, an active metabolite of psilocybinm, is a selective serotonin receptor agonist. Active metabolite of psilocybin. Learn MoreStarting at: $219.00
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Diazoxide
Diazoxide is an antihypertensive, activates ATP-dependent K+ channels (Kir6), which induces activation of PKCε, an intermediate in the opening of mitoKATP channels, results in cardioprotection against hypoxia-induced death. Learn MoreStarting at: $55.00
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TCS 401
TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B) (Ki values are 0.29, 59, 560, 1100, > 2000, > 2000 and > 2000 μM for PTP1B, CD45 D1D2, PTPβ, PTPε D1, SHP-1, PTPα D1 and LAR D1D2 respectively). Learn MoreStarting at: $139.00
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Amiloride hydrochloride
Amiloride hydrochloride is Na+ channel blocker, which defines the I2A-amiloride sensitive and I2B-amiloride insensitive imidazoline binding sites. Learn MoreStarting at: $55.00
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ER 27319 maleate
ER 27319 maleate is a selective inhibitor of Syk kinase which inhibits tyrosine phosphorylation of Syk initiated by the engagement of FcεRI in rat and human mast cells. Results in the abrogation of degranulation, TNF-α production (IC50 = 10 μM) and other related signaling events. Learn MoreStarting at: $98.00
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UB 165 fumarate
UB 165 fumarate is a subtype-selective nicotinic agonist. Full agonist at α3β2- and very weak partial agonist at α4β2- containing nAChRs. Ki values are 0.27, 20 (IC50), 2790 and 990 nM for α4β2, α3, α7 and α1β1δε respectively. Learn MoreStarting at: $179.00
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Ro 32-0432 hydrochloride
Ro 32-0432 hydrochloride is a selective cell-permeable protein kinase C inhibitor, which displays slight selectivity for conventional PKC isoforms over Ca2+ and atypical PKC isoforms; binding affinities for rat isoforms are 9, 28, 31, 37 and 108 nM for PKC's α, βΙ, βΙΙ, γ and ε respectively. Learn MoreStarting at: $140.00
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1-Methylpsilocin
1-Methylpsilocin is a potent and selective 5-HT2C agonist (IC50 values are 12 and 633 nM for 5-HT2C and 5-HT2A receptors respectively) which displays high affinity for the 5-HT2B receptor (Ki = 38 nM) but acts as an inverse agonist. Learn MoreStarting at: $95.00
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EIPA
EIPA is a TRPP3 channel inhibitor (IC50 = 10.5 μM), which inhibits the Na+/H+ exchanger (NHE). Learn MoreStarting at: $65.00
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VU 0255035
VU 0255035 is a highly selective muscarinic M1 antagonist (Ki = 14.87 nM), which targets the M1 orthosteric site and reduces pilocarpine-induced seizures in mice. Learn MoreStarting at: $110.00
