Search results for 'VX 702'
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Starting at: $972.00
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Starting at: $800.00
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Starting at: $800.00
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Starting at: $800.00
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Ipsapirone
Ipsapirone is a selective 5-HT1A receptor agonist with a Ki value of 10 nM. Learn MoreStarting at: $99.00
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WAY 207024 dihydrochloride
WAY 207024 dihydrochloride is a gonadotropin releasing hormone receptor (GnRH-R) antagonist that exhibits potent affinity with IC50 values of 12 and 71 nM for human and rat GnRH receptors respectively. Learn MoreStarting at: $189.00
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1,3-Dipropyl-8-phenylxanthine
1,3-Dipropyl-8-phenylxanthine is a selective A1 adenosine antagonist. Learn MoreStarting at: $95.00
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CBiPES hydrochloride
CBiPES hydrochloride is a selective positive allosteric modulator of the mGlu2 receptor with an IC50 value of 98.2 nM. Learn MoreStarting at: $115.00
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CP 775146
CP 775146 is a selective, high affinity PPARα agonist with Ki values of 24.5 nM for PPARα and >10 μM for PPARβ and PPARγ in vitro). Learn MoreStarting at: $169.00
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SB 216641 hydrochloride
CD 2665 is a selective RARβγ antagonist (KD values are 110, 306 and > 1000 nM for RARγ, RARβ and RARα respectively). Learn MoreStarting at: $145.00
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HI TOPK 032
HI TOPK 032 is a T-LAK-cell-originated protein kinase (TOPK) inhibitor, which exhibits selectivity for TOPK over other MAPKK family members including ERK1, JNK1 and p38. Blocks proliferation of HCT116 colon cancer cells; suppresses tumor growth in a colon cancer xenograft model. Also inhibits Chk1 (IC50 = 9.6 μM). Learn MoreStarting at: $159.00
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INCA-6
INCA-6 is an inhibitor of interaction between calcineurin and its substrate nuclear factor of activated T cells (NFAT); blocks at the substrate recognition site but not at the catalytic site (Kd = 0.8 mM). Learn MoreStarting at: $95.00
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Impentamine dihydrobromide
Impentamine dihydrobromide is a potent and highly selective histamine H3 receptor antagonist (pA2 = 8.4); displays > 30000-fold selectivity over H1 and H2 receptors. Learn MoreStarting at: $99.00
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ABT 702 dihydrochloride
ABT 702 dihydrochloride is a potent non-nucleoside adenosine kinase inhibitor (IC50 = 1.7 nM), selective over other sites of adenosine interaction (A1, A2A and A3 receptors, adenosine transporter and adenosine deaminase). Learn MoreStarting at: $180.00
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SB 204070
SB 204070 is a potent and selective 5-HT4 receptor antagonist (pIC50 = 10.1). Displays >5000-fold selectivity for 5-HT4 over 5-HT1A, 5-HT1D, 5-HT1E, 5-HT2A, 5-HT2C, and 5-HT3 receptors which exhibits anxiolytic activity upon systemic administration in vivo. Learn MoreStarting at: $140.00
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NSC 625987
NSC 625987 is a cyclin-dependent kinase (cdk) 4 inhibitor (IC50 = 0.2 μM at cdk4/cyclin D1) which displays > 500-fold selectivity over cdk2 (IC50 > 100 μM for cdc2/cyclin A, cdk2/cyclin A and cdk2/cyclin E). Learn MoreStarting at: $115.00
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DV 7028 hydrochloride
DV 7028 hydrochloride is a selective 5-HT2A receptor antagonist (Ki = 22 nM for at 5-HT2 receptors). Learn MoreStarting at: $105.00
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(±)-Lauroylcarnitine chloride
(±)-Lauroylcarnitine chloride is a homolog of acetylcarnitine chloride. Learn MoreStarting at: $85.00