Search results for '1150'
-
2'-MeCCPA
2'-MeCCPA is a potent and highly selective agonist at A1 adenosine receptors (Ki values are 3.3, 9580, 37600 and 1150 nM for human recombinant A1, A2A, A2B and A3 receptors respectively), which acts as a full agonist and inhibits forskolin-stimulated adenylyl cyclase activity in rat cortical membranes with an IC50 value of 13.1 nM. Learn MoreStarting at: $189.00
-
CNQX
CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex. Learn MoreStarting at: $95.00
-
SR 16584
SR 16584 is a selective α3β4 nAChR antagonist (IC50 = 10.2 μM), which selectively binds α3β4 over α4β2 and α7 subtypes (Ki values are 0.508, >100 and >100 μM, respectively). Learn MoreStarting at: $125.00
-
NF 110
NF 110 is a high affinity P2X3 receptor antagonist (Ki values are 36, 82 and 4144 nM for P2X3, P2X1 and P2X2 recombinant receptors respectively), which potently inhibits α,β-meATP-evoked desensitizing currents in rat DRG neurons (IC50 = 527 nM), and shows antitumor activity against several tumor types. Learn MoreStarting at: $135.00