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Search results for 'hp'
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Ro 51
Ro 51 is a potent, dual P2X3 and P2X2/3 antagonist (IC50 values are 2 and 5 nM for rP2X3 and hP2X2/3 respectively). Learn MoreStarting at: $129.00
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Meclizine dihydrochloride
Meclizine dihydrochloride is a Human pregnane X receptor (hPXR) agonist; stronger activator of hPXR than rat PXR. Learn MoreStarting at: $55.00
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PHP 501 trifluoroacetate
PHP 501 trifluoroacetate is a potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters. Learn MoreStarting at: $150.00
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CHPG Sodium salt
CHPG Sodium salt is a sodium salt of the selective mGlu5 agonist CHPG. Learn MoreStarting at: $90.00
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MRS 4062 triethylammonium salt
MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively). Learn MoreStarting at: $180.00
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(RS)-4-Carboxy-3-hydroxyphenylglycine
(RS)-4-Carboxy-3-hydroxyphenylglycine is a broad spectrum EAA agonist/antagonist. Learn MoreStarting at: $135.00
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(R)-3-Carboxy-4-hydroxyphenylglycine
(R)-3-Carboxy-4-hydroxyphenylglycine is a moderately potent NMDA and AMPA/kainate receptor antagonist. Learn MoreStarting at: $280.00
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(RS)-3,5-DHPG
(RS)-3,5-DHPG is a selective group I metabotropic glutamate receptor agonist which activates both mGlu1 and mGlu5. Learn MoreStarting at: $49.00
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m-3M3FBS
m-3M3FBS is a activator of phospholipase C (PLC), which stimulates superoxide generation, Ca2+ release and inositol phosphate formation in a variety of cell types, and inhibits growth of the leukemic cell lines U937 and THP-1. Learn MoreStarting at: $98.00
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NPE-caged-HPTS
NPE-caged-HPTS is a caged fluorescent pH indicator. Learn MoreStarting at: $199.00
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AZ 11645373
AZ 11645373 is a potent and selective human P2X7 antagonist (KB values are 5 - 7 and > 10,000 nM at hP2X7 and rP2X7 respectively) that is completely without effect at all other P2X subtypes. Learn MoreStarting at: $140.00
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TCS 401
TCS 401 is a selective inhibitor of protein-tyrosine phosphatase 1B (PTP1B) (Ki values are 0.29, 59, 560, 1100, > 2000, > 2000 and > 2000 μM for PTP1B, CD45 D1D2, PTPβ, PTPε D1, SHP-1, PTPα D1 and LAR D1D2 respectively). Learn MoreStarting at: $139.00
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Ciliobrevin A
Ciliobrevin A is a hedgehog (Hh) pathway antagonist which blocks Sonic hedgehog (Shh)-induced Hh pathway activation (IC50 = 7 μM) downstream of Smo. Learn MoreStarting at: $119.00
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2-ThioUTP tetrasodium salt
2-ThioUTP tetrasodium salt is a potent and selective P2Y2 agonist (EC50 values are 0.035, 0.35 and 1.5 μM for hP2Y2, hP2Y4 and hP2Y6 receptors respectively). Learn MoreStarting at: $269.00
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ACHP
ACHP is a IκB kinase inhibitor (IC50 values are 8.5 and 250 nM for IKKβ and IKKα respectively), which inhibits DNA binding activity of NF-κB. Blocks NF-κB pathway in multiple myeloma cell lines; induces cell growth arrest and apoptosis. Learn MoreStarting at: $209.00
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CDP 840 hydrochloride
(S)-3,5-DHPG is a selective group I mGlu receptor agonist. Learn MoreStarting at: $135.00
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(S)-3,5-DHPG
BYK 49187 is a PARP-1 and PARP-2 inhibitor (pIC50 values are 8.36 and 7.50 for cell-free recombinant PARP-1 and murine PARP-2 respectively) which displays potent inhibitory activity against human PARP-1 in cell-free and cellular assays in vitro. Learn MoreStarting at: $95.00
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SC 236
CHPG is a selective mGlu5 metabotropic glutamate receptor agonist, completely inactive at mGlu1a receptors expressed in CHO cells. Learn MoreStarting at: $110.00
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CHPG
E4CPG is a novel group I/group II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG. Learn MoreStarting at: $80.00
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Allopregnanolone
Allopregnanolone is GABAA receptor positive allosteric modulator. Learn More
