Search results for 'ganoderic acid'
-
3,5-DHBA
3,5-DHBA is a selective agonist of hydroxycarboxylic acid receptor 1 (HCA1, also known as GPR81) (EC50 ~150 μM), Inhibits lipolysis in wild-type mouse adipocytes. Learn MoreStarting at: $59.00
-
Kynurenic acid sodium salt
Kynurenic acid sodium salt is a sodium salt of kynurenic acid, and it is a broad spectrum EAA antagonist. Learn MoreStarting at: $79.00
-
Valerenic acid
Valerenic acid is a positive allosteric modulator of GABAA receptors, which wdisplays preference for receptors containing β2 or β3 subunits and activates the receptor and also blocks the channel at high concentrations. Learn MoreStarting at: $85.00
-
22-Oxacalcitriol
22-Oxacalcitriol is non-calcemic vitamin D3 analog and VDR ligand, which inhibits tumor growth of osteosarcoma in vitro in combination with all-trans retinoic acid. Learn MoreStarting at: $125.00
-
TUG 424
TUG 424 is an agonist of the free fatty acid receptor FFA1 (GPR40) (EC50 = 32 nM), which enhances glucose-stimulated insulin secretion in INS-1E cells at 100 nM. Learn MoreStarting at: $110.00
-
Ch 55
Ch 55 is a highly potent synthetic retinoid that has high affinity for RAR-α and RAR-β receptors and low affinity for cellular retinoic acid binding protein (CRABP) and Inhibits rabbit tracheal epithelial cell differentiation by inhibiting transglutaminase and increasing cholesterol sulfate (EC50 values are 0.02 and 0.03 nM respectively). Learn MoreStarting at: $90.00
-
L-Cysteinesulfinic acid
L-Cysteinesulfinic acid is a agonist at mGlu1a and mGlu5a subtypes expressed in clonal RGT cell lines. Also agonist at NMDA and PLD-coupled mGlu receptors. Learn MoreStarting at: $70.00
-
cis-Ned 19
cis-Ned 19 is an irreversible nicotinic acid adenine dinucleotide phosphate (NAADP) antagonist, which inhibits Ca2+ release (IC50 = 800 nM) and [32P]NAADP binding (IC50 = 15 μM). Learn MoreStarting at: $195.00
-
5,7-Dichlorokynurenic acid sodium salt
Sodium salt of 5,7-Dichlorokynurenic acid, a potent antagonist at the glycine site of the NMDA receptor (Ki = 79 nM vs. [3H]-glycine). Learn MoreStarting at: $65.00
-
(-)-Terreic acid
Selective inhibitor of Bruton's tyrosine kinase (BTK), which inhibits the interaction between PKCbII and BTK (IC50 ~ 30 mM) and the catalytic activity of BTK but does not affect the activity of PKC. Learn MoreStarting at: $155.00
-
MNI-caged-NMDA
MNI-caged-NMDA is a NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $175.00
-
7-Chlorokynurenic acid sodium salt
7-Chlorokynurenic acid sodium salt is a sodium salt of 7-Chlorokynurenic acid, an NMDA receptor antagonist acting at the glycine site. Learn MoreStarting at: $65.00
-
N-ArachidonylGABA
N-ArachidonylGABA is a arachidonyl amino acid; first isolated from bovine brain. Learn MoreStarting at: $80.00
-
TC-F 2
TC-F 2 is a potent, reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 values are 28 and 100 nM for human and rat FAAH respectively), which displays selectivity for FAAH over cannabinoid-related targets (IC50 > 20 μM for CB1, CB2 and TRPV1). Learn MoreStarting at: $155.00
-
5,7-Dichlorokynurenic acid
5,7-Dichlorokynurenic acid is a potent antagonist at the glycine site of the NMDA receptor (Ki = 79 nM vs. [3H]-glycine). Learn MoreStarting at: $65.00
-
MNI caged kainic acid
MNI caged kainic acid is a kainic acid caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $350.00
-
NCS-382
NCS-382 is a γ-Hydroxybutyric acid antagonist, anticonvulsant. Learn MoreStarting at: $80.00
-
CCMQ
CCMQ is used in conjunction with [3H]-homoquinolinic acid to characterize NR2B-containing NMDA receptors which selectively inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites. Learn MoreStarting at: $95.00
-
Ethacrynic acid - d5
Ethacrynic acid - d5 is a deuterated ethacrynic acid which used as an internal standard for GC- or LC-mass spectrometry. Learn MoreStarting at: $105.00
-
SA 57
SA 57 is a potent inhibitor of fatty acid amide hydrolase (FAAH) (IC50 < 10 nM), which inhibits both human and mouse FAAH enzymes and displays inhibitory activity against FAAH, MAGL and ABHD6 in vivo. Learn MoreStarting at: $100.00