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Search results for 'PI 103'
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Spironolactone
Spironolactone is a competitive mineralocorticoid (aldosterone) receptor antagonist that exhibits antihypertensive activity in vivo, displays antiandrogen activity and inhibits steroid hormone biosynthesis. Learn MoreStarting at: $45.00
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Caffeine
Caffeine is a central nervous system stimulant, which mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors. Learn MoreStarting at: $69.00
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m-Chlorophenylbiguanide hydrochloride
m-Chlorophenylbiguanide hydrochloride is a prototypical potent and selective 5-HT3 receptor agonist. Learn MoreStarting at: $69.00
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(±)-Acetylcarnitine chloride
(±)-Acetylcarnitine chloride is weak cholinergic agonist and important intermediates in lipid metabolism. Learn MoreStarting at: $49.00
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SU 4312
SU 4312 is a potent and selective inhibitor of VEGFR and PDGFR tyrosine kinases (IC50 values are 0.8 and 19.4 μM respectively). Learn MoreStarting at: $189.00
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Sodium citrate
Sodium citrate is commonly used laboratory reagent Learn MoreStarting at: $39.00
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DHBP dibromide
DHBP dibromide is a blocks calcium release from sarcoplasmic reticulum by direct interaction with the ryanodine receptor. Learn MoreStarting at: $55.00
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Pentoxifylline
Pentoxifylline is a phosphodiesterase inhibitor that blocks production of TNF-&alpha and other cytokines. Learn MoreStarting at: $69.00
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(±)-Lauroylcarnitine chloride
(±)-Lauroylcarnitine chloride is a homolog of acetylcarnitine chloride. Learn MoreStarting at: $85.00
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AS 19
AS 19 is a potent 5-HT7 receptor agonist (IC50 = 0.83 nM), that enhances memory consolidation and reverses scopolamine- or dizocilpine-induced amnesia in vivo. Learn MoreStarting at: $109.00
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1-EBIO
1-EBIO is an activator of epithelial KCa channels, stimulates a large and sustained trans-epithelial Cl- secretory response across T84 monolayers. And it also induces hyperpolarization to the same magnitude as ACh in aortic value endothelial cells. Learn MoreStarting at: $65.00
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PF 04691502
PF 04691502 is an potent and selective dual ATP-competitive PI 3-K/mTOR inhibitor (Ki values are 1.6, 1.8, 1.9, 2.1 and 16 nM for human PI 3-K δ, α, γ, β, and mTOR, respectively). Learn MoreStarting at: $145.00
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Jasplakinolide
Jasplakinolide Rapidly stabilizes pre-formed actin filaments and inhibits their disassembly in vitro.It also induces polymerization of actin monomers into F-actin in vivo. Learn MoreStarting at: $205.00
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RO-3
RO-3 is a selective homomeric P2X3 and heteromeric P2X2/3 receptor antagonist (pIC50 values are 7.0 and 5.9 respectively) that exhibits no activity at P2X1, P2X2, P2X4, P2X5 and P2X7 receptors (IC50 > 10 μM). Learn MoreStarting at: $105.00
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L-655,240
L-655,240 is a potent and selective thromboxane A2/prostaglandin endoperoxide receptor antagonist. pA2 values are 8 - 8.4 in guinea pig smooth muscle; IC50 = 7 nM for inhibition of human platelet aggregation. Orally active in vivo. Learn MoreStarting at: $105.00
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Taltirelin
Taltirelin is a synthetic thyrotropin-releasing hormone (TRH) analog which displays ~ 30 - 100-fold more potent CNS activity and ~ 50-fold weaker endocrine activity than TRH. Learn MoreStarting at: $69.00
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L-364,373
L-364,373 is a activator of KV7.1 (KCNQ1) channels. Learn MoreStarting at: $140.00
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Devazepide
Devazepide is a potent, orally active CCK1 (CCK-A) receptor antagonist that displays appetite-stimulant effects. Devazepide blocks the anorectic response to CCK-8 and increases food intake in rats following systemic and i.c.v administration. Learn MoreStarting at: $149.00
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Z-Cyclopentyl-AP4
Z-Cyclopentyl-AP4 is a group III mGlu receptor agonist that exhibits higher potency at mGlu4 than mGlu8 (EC50 values are 49 and 124 μM respectively) with no activity at mGlu7. And selectively inhibits synaptic activity in the lateral perforant pathway (IC50 values are 130 and 1859 μM in the lateral and medial perforant pathways respectively). Learn MoreStarting at: $129.00
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D-myo-Inositol 1,4,5-trisphosphate, hexapotassium salt
D-myo-Inositol 1,4,5-trisphosphate, hexapotassium salt, as an important second messenger involved in Ca2+ mobilization from intracellular stores (EC50 = 0.1 μM), is formed from the enzymatic hydrolysis of phosphatidyl inositol-4,5-bisphosphate. . Learn MoreStarting at: $119.00
