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Search results for 'Glutamate'
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Chicago Sky Blue 6B
Chicago Sky Blue 6B is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits macrophage migration inhibitory factor (MIF) (IC50 = 0.81 μM) and MIF proinflammatory activity. Learn MoreStarting at: $49.00
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Ceftriaxone disodium salt
Ceftriaxone disodium salt is β-lactam antibiotic, which increased activity of the EAAT2 glutamate transporter and displays neuroprotective activity in vivo via upregulation. Learn MoreStarting at: $49.00
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2,4-Dihydroxyphenylacetyl-L-asparagine
2,4-Dihydroxyphenylacetyl-L-asparagine is a constituent of various spider toxins. Which has been reported to be specific blocker of glutamate receptors. Learn MoreStarting at: $135.00
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Lamotrigine isethionate
Lamotrigine isethionate is a water-soluble salt of lamotrigine, and displays anticonvulsant effects and inhibits glutamate release, possibly through inhibition of Na+, K+ and Ca2+ currents. Learn MoreStarting at: $90.00
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L-CCG-l
L-CCG-l is a potent group II metabotropic glutamate receptor agonist. Learn MoreStarting at: $185.00
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L-CCG-lll
L-CCG-lll is a potent and competitive inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate. Learn MoreStarting at: $265.00
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(RS)-PPG
(RS)-PPG is a potent and selective group III metabotropic glutamate receptor agonist, with approximately 25-fold preference for hmGlu8. Learn MoreStarting at: $100.00
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MFZ 10-7
MFZ 10-7 is a high affinity negative allosteric modulator at the mGlu5 receptor (Ki = 0.67 nM), which potently inhibits mGlu5 glutamate-mediated calcium mobilization (IC50 = 1.22 nM). Learn MoreStarting at: $105.00
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(RS)-MCPG disodium salt
(RS)-MCPG disodium salt is a sodium salt of (RS)-MCPG, a non-selective group I/group II metabotropic glutamate receptor antagonist. Learn MoreStarting at: $95.00
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Sipatrigine
Sipatrigine is a blocker of voltage-dependent sodium channels (NaV) which inhibits glutamate release and displays neuroprotective activity in rat models of cerebral ischemia. Learn MoreStarting at: $145.00
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(S)-4-Carboxyphenylglycine
(S)-4-Carboxyphenylglycine is a competitive group I metabotropic glutamate receptor antagonist, with selectivity for mGlu1a/1a over mGlu5a/5b. Learn MoreStarting at: $135.00
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Pentamidine isethionate
Antimicrobial. Neuroprotective; inhibits constitutive nitric oxide synthase in the brain and acts as a NMDA glutamate receptor antagonist. Learn MoreStarting at: $80.00
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(RS)-MCPG
(RS)-MCPG is a non-selective group I/group II metabotropic glutamate receptor antagonist. Learn MoreStarting at: $95.00
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CGP 55845 hydrochloride
CGP 55845 hydrochloride is a potent, selective GABAB receptor antagonist (IC50 = 5 nM) that prevents agonist binding (pKi = 8.35) and inhibits GABA and glutamate release (pEC50 values are 8.08 and 7.85 respectively). Learn MoreStarting at: $140.00
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(S)-MCPG
(S)-MCPG is a active isomer of (RS)-MCPG. Non-selective group I/group II metabotropic glutamate receptor antagonist. Learn MoreStarting at: $185.00
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DFB
DFB is a novel allosteric potentiator of the metabotropic glutamate receptor mGlu5. Learn MoreStarting at: $70.00
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PMPA (NAALADase inhibitor)
PMPA (NAALADase inhibitor) is a highly potent and selective inhibitor of glutamate carboxypeptidase 2 (GCP II/N-acetylated α-linked dipeptidase/NAALADase) with a Ki value of 275 pM. Learn MoreStarting at: $90.00
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7-Chlorokynurenic acid
7-Chlorokynurenic acid is a NMDA receptor antagonist acting at the glycine site. Potent competitive inhibitor of L-glutamate transport into synaptic vesicles. Learn MoreStarting at: $60.00
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(RS)-3,5-DHPG
(RS)-3,5-DHPG is a selective group I metabotropic glutamate receptor agonist which activates both mGlu1 and mGlu5. Learn MoreStarting at: $49.00
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DL-AP3
DL-AP3 is a competitive group I metabotropic glutamate receptor antagonist and inhibitor of phosphoserine phosphatase. Learn MoreStarting at: $75.00
