Search results for 'AG 490'
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Pronethalol hydrochloride
Pronethalol hydrochloride is a ??-adrenergic antagonist, clinically effective in the treatment of angina pectoris and some arrhythmias. Learn MoreStarting at: $69.00
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Spironolactone
Spironolactone is a competitive mineralocorticoid (aldosterone) receptor antagonist that exhibits antihypertensive activity in vivo, displays antiandrogen activity and inhibits steroid hormone biosynthesis. Learn MoreStarting at: $45.00
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Prochlorperazine dimaleate
Prochlorperazine dimaleate is a D2 receptor antagonist. Learn MoreStarting at: $55.00
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3,5-DHBA
3,5-DHBA is a selective agonist of hydroxycarboxylic acid receptor 1 (HCA1, also known as GPR81) (EC50 ~150 μM), Inhibits lipolysis in wild-type mouse adipocytes. Learn MoreStarting at: $59.00
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m-Chlorophenylbiguanide hydrochloride
m-Chlorophenylbiguanide hydrochloride is a prototypical potent and selective 5-HT3 receptor agonist. Learn MoreStarting at: $69.00
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Kynurenic acid sodium salt
Kynurenic acid sodium salt is a sodium salt of kynurenic acid, and it is a broad spectrum EAA antagonist. Learn MoreStarting at: $79.00
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(±)-Acetylcarnitine chloride
(±)-Acetylcarnitine chloride is weak cholinergic agonist and important intermediates in lipid metabolism. Learn MoreStarting at: $49.00
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Chicago Sky Blue 6B
Chicago Sky Blue 6B is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits macrophage migration inhibitory factor (MIF) (IC50 = 0.81 μM) and MIF proinflammatory activity. Learn MoreStarting at: $49.00
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DL-Dithiothreitol
DL-Dithiothreitol is a reagent for maintaining SH groups in the reduced state. Learn MoreStarting at: $119.00
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Sodium citrate
Sodium citrate is commonly used laboratory reagent Learn MoreStarting at: $39.00
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AS 19
AS 19 is a potent 5-HT7 receptor agonist (IC50 = 0.83 nM), that enhances memory consolidation and reverses scopolamine- or dizocilpine-induced amnesia in vivo. Learn MoreStarting at: $109.00
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VUF 8430 dihydrobromide
VUF 8430 dihydrobromide is a high affinity (pKi = 7.5), potent histamine H4 receptor full agonist (pEC50 = 7.3). Displays moderate affinity for H3 receptors (pKi = 6.0) and weak partial agonist activity at H2 receptors. Learn MoreStarting at: $109.00
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CPT 11
CPT 11 is an inhibitor of DNA topoisomerase I that displays antitumor activity against a range of tumor types. Learn MoreStarting at: $139.00
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Calcium chloride dihydrate
Calcium chloride dihydrate is a commonly used laboratory reagent Learn MoreStarting at: $79.00
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1-EBIO
1-EBIO is an activator of epithelial KCa channels, stimulates a large and sustained trans-epithelial Cl- secretory response across T84 monolayers. And it also induces hyperpolarization to the same magnitude as ACh in aortic value endothelial cells. Learn MoreStarting at: $65.00
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NF 546
NF 546 is a P2Y11 agonist (pEC50 = 6.27). Exhibits selectivity for P2Y11 over a range of P2Y and P2X receptors. Learn MoreStarting at: $149.00
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(RS)-CPP
(RS)-CPP is a potent NMDA antagonist. Separate isomer (R)-CPP also available. Learn MoreStarting at: $129.00
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CY 208-243
CY 208-243 is a centrally active dopamine D1 receptor agonist, selective over D2 receptor sites, which stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM, that exerts antiParkinsonian activity in animal models. Learn MoreStarting at: $139.00
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MRS 2179 tetrasodium salt
MRS 2179 tetrasodium salt is a competitive antagonist at P2Y1 receptors (KB = 100 nM). Learn MoreStarting at: $145.00
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Gadolinium chloride
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist and induces NLRP3 inflammasome activation in bone marrow-derived macrophages. Learn MoreStarting at: $39.00