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Search results for 'ganoderic acid'
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(±)-HIP-A
(±)-HIP-A is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.6 μM) rather than [3H]L-glutamate uptake (IC50 = 18 μM). Learn MoreStarting at: $139.00
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(±)-HIP-B
(±)-HIP-B is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.2 μM) rather than [3H]L-glutamate uptake (IC50 = 16.9 μM). Learn MoreStarting at: $139.00
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2-Palmitoylglycerol
2-Palmitoylglycerol is an endogenous fatty acid glycerol ester that enhances activity of 2-arachidonylglycerol. Learn MoreStarting at: $55.00
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trans-4-Hydroxycrotonic acid
trans-4-Hydroxycrotonic acid binds to the γ-hydroxybutyric acid (GHB) receptor with higher affinity than GHB itself. Learn MoreStarting at: $90.00
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AM 1172
AM 1172 metabolically stable anandamide uptake inhibitor (IC50 = 2.1 - 2.5 μM) and fatty acid amide hydrolase (FAAH) inhibitor (Ki = 3.18 μM). Learn MoreStarting at: $139.00
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BMS 195614
BMS 195614 is a neutral retinoic acid receptor (RAR) α-selective antagonist (Ki = 2.5 nM) which displays no significant effect on nuclear receptor corepressor (NCoR) binding; moderately decreases SMRT binding to RAR. Learn MoreStarting at: $159.00
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CID 2745687
CID 2745687 is a competitive, reversible antagonist of the orphan receptor GPR35 (Ki = 12.8 nM) which blocks the GPR35-mediated increase in ERK1/2 phosphorylation and β-arrestin recruitment induced by pamoic acid. Learn MoreStarting at: $119.00
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Hypotaurine
Endogenous inhibitory amino acid. Learn MoreStarting at: $75.00
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4-CMTB
4-CMTB is a free fatty acid receptor FFA2 agonist (pEC50 = 6.38) and positive allosteric modulator, which binds at a site distinct from the orthosteric site; modulates the activity of short-chain fatty acids at FFA2 via the FFA2 second extracellular loop (ECL2). Learn MoreStarting at: $105.00
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Homovanillic acid
Homovanillic acid is a fluorimetric reagent and major catecholamine metabolite, which has been used for fluorimetric determination of oxidative enzymes including glucose oxidase. Learn MoreStarting at: $49.00
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Spaglumic acid
Spaglumic acid is the most abundant peptide neurotransmitter in the mammalian CNS. Learn MoreStarting at: $109.00
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1-Oleoyl lysophosphatidic acid sodium salt
1-Oleoyl lysophosphatidic acid sodium salt is an endogenous agonist of the lysophospholipid receptors LPA1 and LPA2, which inhibits differentiation of neural stem cells (NSCs) into neurons. Learn MoreStarting at: $45.00
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GRI 977143
GRI 977143 is a selective lysophosphatidic acid 2 (LPA2) receptor non-lipid agonist (EC50 = 3.3 μM), which inhibits activation of caspases 3, 7, 8 and 9, Bax translocation and PARP-1 cleavage. Learn MoreStarting at: $135.00
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HexylHIBO
HexylHIBO is a group I mGlu receptor antagonist (Ki values are 140 and 110 μM at mGlu1a and mGlu5a receptors respectively), which decreases sEPSCs in rat pyramidal neurons in vitro. Learn MoreStarting at: $129.00
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(S)-HexylHIBO
(S)-HexylHIBO is a group I mGlu receptor antagonist (Kb values are 30 and 61 μM at mGlu1a and mGlu5a receptors respectively). Learn MoreStarting at: $139.00
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BCTC
BCTC is an orally effective vanilloid receptor 1 (TRPV1 receptor) antagonist, which inhibits acid- and capsaicin-induced activation of rat TRPV1 receptors (IC50 values are 6.0 and 35 nM respectively). Learn MoreStarting at: $109.00
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H2L 5765834
Antagonist of the lysophosphatidic acid receptors LPA1, LPA5 and LPA3 (IC50 values are 94, 463 and 752 nM respectively). Learn MoreStarting at: $139.00
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SB 452533
SB 452533 is a potent TRPV1 antagonist against capsaicin (pKb = 7.7), noxious heat and acid-mediated (pIC50 = 7.0) receptor activation (pKi = 6.22 at the recombinant hTRPV1 receptor). Learn MoreStarting at: $109.00
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Kainic acid
Kainic acid is a selective agonist at kainate receptors. Potent excitant and neurotoxin. Learn MoreStarting at: $65.00
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Homoquinolinic acid
Homoquinolinic acid is a potent NMDA receptor agonist; subtype-selective. Learn MoreStarting at: $129.00
