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Search results for 'ganoderic acid'
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trans-Ned 19
trans-Ned 19 is a nicotinic acid adenine dinucleotide phosphate (NAADP) antagonist, which inhibits NAADP-mediated Ca2+ release (IC50 = 6 nM) and [32P]NAADP binding (IC50 = 0.4 nM). Learn MoreStarting at: $210.00
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N-Acetylglycyl-D-glutamic acid
N-Acetylglycyl-D-glutamic acid is an excitatory peptide, more potent than L-glutamic acid at inducing seizures in mice. Learn MoreStarting at: $80.00
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PALDA
PALDA is an endogenous fatty acid dopamide that displays 'entourage' effects on endovanilloids NADA and anandamide. Learn MoreStarting at: $75.00
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H2L5186303
H2L5186303 is a potent and selective lysophosphatidic acid 2 (LPA2) receptor antagonist (IC50 values are 8.9, 1230 and 27354 nM for LPA2, LPA3 and LPA1 receptors respectively, in a LPA-elicited calcium mobilization assay). Learn MoreStarting at: $135.00
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Domoic acid
Domoic acid is more potent and possibly more selective than kainate at kainate receptors, as demonstrated in electrophysiological studies. Learn MoreStarting at: $110.00
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L-703,664 succinate
L-703,664 succinate is a 5-HT1D receptor agonist that displays selectivity over other 5-HT receptor subtypes (pIC50 values are 7.2, 6.1, < 5.0 and < 5.0 for 5-HT1D, 5-HT1A, 5-HT2A and 5-HT3 respectively) and other receptors (pIC50 < 5.0 for adenosine, adrenergic, excitatory amino acids, dopamine, histamine, muscarinic, nicotinic and opiate receptors). Learn MoreStarting at: $140.00
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Telenzepine dihydrochloride
Telenzepine dihydrochloride is a selective high affinity muscarinic M1 receptor antagonist (Ki = 0.94 nM) which inhibits gastric acid secretion. Learn MoreStarting at: $50.00
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WIN 18446
WIN 18446 is an inhibitor of aldehyde dehydrogenase 1a2 (ALDH1a2) (IC50 = 0.3 μM) which inhibits the biosynthesis of retinoic acid from retinol in neonatal and adult murine testis. Learn MoreStarting at: $80.00
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AACOCF3
AACOCF3 is an inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Learn MoreStarting at: $65.00
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LE 135
LE 135 is a retinoic acid antagonist; displays moderate selectivity for RARβ over RARα Learn MoreStarting at: $105.00
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D-Aspartic acid
Endogenous NMDA receptor agonist with similar activity to the L-isomer (L-aspartic acid). Learn MoreStarting at: $80.00
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7-Chlorokynurenic acid
7-Chlorokynurenic acid is a NMDA receptor antagonist acting at the glycine site. Potent competitive inhibitor of L-glutamate transport into synaptic vesicles. Learn MoreStarting at: $60.00
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DLPC
DLPC is a selective agonist of the orphan nuclear receptor LRH-1 (liver receptor homolog-1, NR5A2) in vitro, which induces bile acid biosynthetic enzymes; increases bile acid and decreases hepatic triglycerides and serum glucose, and exhibits antidiabetic effects. Learn MoreStarting at: $50.00
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Arachidonyl serotonin
Arachidonyl serotonin is a dual fatty acid amide hydrolase (FAAH) inhibitor/TRPV1 antagonist (IC50 values are 5.6 μM and 37 - 40 nM for FAAH and TRPV1 respectively). Learn MoreStarting at: $75.00
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MAFP
MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). It also binds irreversibly to CB1 receptors (IC50 = 20 nM). Learn MoreStarting at: $98.00
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Palmitoylisopropylamide
Palmitoylisopropylamide is an inhibitor of fatty acid amide hydrolase (FAAH); pIC50 = 4.89 for inhibition of [3H]-anandamide metabolism. Learn MoreStarting at: $65.00
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C 75
C 75 is a synthetic inhibitor of fatty acid synthase (FAS) which inhibits fatty acid synthesis in vitro and in vivo and displays anorectic effects. Induces apoptosis in MCF-7 xenografts and exhibits anti-tumor activity. Learn MoreStarting at: $135.00
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Rosmarinic acid
Rosmarinic acid is an anti-inflammatory, cytostatic and antiviral, which also displays agonist activity at GPR35. Learn MoreStarting at: $95.00
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DL-TBOA
DL-TBOA is a competitive, non-transportable blocker of excitatory amino acid transporters (IC50 values are 70, 6, and 6 μM for EAAT1, EAAT2 and EAAT3 respectively), which also inhibits EAAT4 and EAAT5 (Ki values are 4.4 and 3.2 μM respectively). Learn MoreStarting at: $140.00
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BMS 493
BMS 493 is a pan-retinoic acid receptor (pan-RAR) inverse agonist, which enhances nuclear corepressor (NCoR) interaction with RARs. Learn MoreStarting at: $135.00
