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Search results for 'WIN'
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PF 514273
PF 514273 is a potent and selective CB1 receptor antagonist that inhibits food intake in vivo following oral administration. Learn MoreStarting at: $139.00
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(R)-(+)-8-Hydroxy-DPAT hydrobromide
(R)-(+)-8-Hydroxy-DPAT hydrobromide is a full 5-HT1A serotonin receptor agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. It is more active enantiomer of 8-Hydroxy-DPAT hydrobromide. Learn MoreStarting at: $109.00
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8-Hydroxy-DPAT hydrobromide
8-Hydroxy-DPAT hydrobromide is a standard selective 5-HT1A agonist that reduces hippocampal 5-HT levels following systemic administration in rats in vivo. Learn MoreStarting at: $59.00
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WAY 161503 hydrochloride
WAY 161503 hydrochloride is a potent and selective 5-HT2C receptor agonist with antidepressant effect following systemic administration in vivo. Learn MoreStarting at: $99.00
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Remoxipride hydrochloride
Remoxipride hydrochloride is a dopamine D2 receptor antagonist showing selectivity over D3 and D4 receptors with Ki values of ~ 300, ~ 1600, and ~ 2800 nM for D2, D3 and D4 receptors respectively. Learn MoreStarting at: $105.00
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UK 14304
UK 14304 is a full α2 adrenergic agonist that is centrally active following systemic administration in vivo. Learn MoreStarting at: $89.00
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Ticlopidine hydrochloride
Ticlopidine hydrochloride, a selective P2Y12 receptor antagonist, inhibits ADP-induced platelet aggregation and displays antithrombotic activity following oral administration in vivo. Learn MoreStarting at: $38.00
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CV 1808
CV 1808, a adenosine A2 receptor agonist, is coronary vasodilator, antihypertensive and antipsychotic following systemic administration in vivo. Learn MoreStarting at: $65.00
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MPPG
MTPG is a group II/group III metabotropic glutamate receptor antagonist, showing selectivity for group II in electrophysiological studies. Learn MoreStarting at: $135.00
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MSPG
MPPG is a potent antagonist of L-AP4-induced effects in rat spinal cord, thalamic and hippocampal neurons, showing selectivity over (1S,3S)-ACPD-induced effects. Potent antagonist of mGlu receptors linked to adenylyl cyclase in adult rat cortical slices. Learn MoreStarting at: $135.00
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MAP4
(S)-SNAP 5114 is a GABA transport inhibitor, showing selectivity for GAT-3 and GAT-2 (IC50 values are 5, 21 and 388 μM for hGAT-3, rGAT-2 and hGAT-1 respectively). Learn MoreStarting at: $135.00
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BMS 470539 dihydrochloride
BMS 470539 dihydrochlorideis a potent, selective melanocortin MC1 receptor agonist (IC50 = 120 nM), which exhibits anti-inflammatory properties following ischemia-reperfusion in the vasculature. Learn MoreStarting at: $169.00
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Burimamide oxalate
Burimamide oxalate is a histamine H3/H2 receptor antagonist (Ki values are 0.07, 7.8 and 290 μM for H3, H2 and H1 receptors respectively), which displays partial agonist activity in SK-N-MC cells and produces antinociceptive effects following intraventricular administration (ED50 = 183 nmol/mouse in hot-plate test). Learn MoreStarting at: $115.00
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Bay 36-7620
Bay 36-7620 is a selective mGlu1 receptor non-competitive antagonist (IC50 = 0.16 μM) with inverse agonist activity, which exhibits neuroprotective and anticonvulsive effects in vivo following systemic administration. Learn MoreStarting at: $155.00
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AM 281
AM 281 is a potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively), which increases locomotor activity following systemic administration in vivo. Learn MoreStarting at: $140.00
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(S)-3,4-DCPG
(S)-3,4-DCPG is a potent, selective mGlu8a agonist (EC50 = 31 nM). Displays > 100-fold selectivity over mGlu1-7, which increases c-Fos expression in stress-related brain areas following systemic administration in mice in vivo. Learn MoreStarting at: $140.00
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SNC 162
SNC 162 is a potent and selective non-peptide δ-opioid receptor agonist (Ki = 0.63 nM) which displays > 8000-fold selectivity over μ-opioid receptors and is centrally active following systemic administration in vivo. Learn MoreStarting at: $160.00
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BMS 182874 hydrochloride
BMS 182874 hydrochloride is a potent, selective and competitive non-peptide endothelin ETA receptor antagonist (Ki = 48 nM) which displays > 1000-fold selectivity over ETB receptors. Inhibits ET-1-induced pressor response following oral or intravenous administration in vivo and inhibits ET-1-induced longitudinal muscle contraction in the mouse colon in vitro. Learn MoreStarting at: $140.00
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WIN 64338 hydrochloride
L-NIL hydrochloride is the first potent, non-peptide, competitive bradykinin B2 receptor antagonist. Learn MoreStarting at: $110.00
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A 77636 hydrochloride
A 77636 hydrochloride is a potent and selective dopamine D1-like receptor agonist (pEC50 values are 8.97 and < 5 for D1-like and D2-like receptors respectively), which displays anti-Parkinsonian activity following oral administration in vivo. Learn MoreStarting at: $140.00
