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Search results for 'PI'
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Anti-PIKFyve
Anti-PIKFyve is an antibody raised against recombinant protein corresponding to amino acid residues 1083-1200 of human PIKfyve . Learn MoreStarting at: $299.00
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MRS 2211
MRS 2211 is a competitive P2Y13 receptor antagonist (pIC50 = 5.97) that displays > 20-fold selectivity over P2Y1 and P2Y12 receptors. Learn MoreStarting at: $89.00
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Ro 19-4603
Ro 19-4603 is a benzodiazepine inverse agonist, which binds with high affinity to both diazepam-sensitive (DS) and diazepam-insensitive (DI) GABAA receptors (Ki values are ~ 0.2 and ~ 2.6 nM for DS and DI receptors respectively). Learn MoreStarting at: $99.00
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Anpirtoline hydrochloride
Anpirtoline hydrochloride is a highly potent 5-HT1B receptor agonist (Ki values are 28, 150 and 1490 nM at 5-HT1B, 5-HT1A and 5-HT2 receptors respectively), which decreases central serotonin synthesis and attenuates aggressive behavior in vivo. It also acts as an antagonist at 5-HT3 receptors (Ki = 29.5 nM) and is brain penetrant. Learn MoreStarting at: $119.00
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Fentanyl citrate
Fentanyl citrate is a potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively), which displays antinociceptive activity in vivo. Learn MoreStarting at: $55.00
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Ipsapirone
Ipsapirone is a selective 5-HT1A receptor agonist with a Ki value of 10 nM. Learn MoreStarting at: $99.00
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CYM 5541
CYM 5541 is a selective sphingosine-1-phosphate receptor 3 (S1P3) allosteric agonist that occupies a different space within the ligand binding pocket of S1P3 than S1P. Learn MoreStarting at: $115.00
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ZAPA sulfate
ZAPA sulfate is a useful ligand to investigate GABA receptors linked to benzodiazepine receptors. It is also a GABAC receptor antagonist. Learn MoreStarting at: $95.00
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Ro 15-4513
Ro 15-4513 is a high affinity benzodiazepine ligand that acts as partial inverse agonist at recombinant DS α1-, α2-, α3- and α5-GABAA receptors. Learn MoreStarting at: $115.00
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AC 55541
AC 55541 is a potent and selective protease-activated receptor 2 (PAR2) agonist that stimulates cell proliferation, PI hydrolysis and Ca2+ mobilization in vitro and exhibits pronociceptive activity in vivo. Learn MoreStarting at: $149.00
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Ropinirole
Ropinirole is a selective D2-like receptor agonist (D3 > D2 > D4). Learn MoreStarting at: $55.00
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W146
W146 is a potent sphingosine-1-phosphate receptor S1P1 selective antagonist that enhances capillary leakage and restores lymphocyte egress in vivo. Learn MoreStarting at: $109.00
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BF 2649 hydrochloride
BF 2649 hydrochloride is a histamine H3 receptor inverse agonist and antagonist that exhibits nootropic effects in cognitive disorders; reduces locomotor hyperactivity induced by methamphetamine. Learn MoreStarting at: $105.00
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(±)-Clopidogrel hydrochloride
(±)-Clopidogrel hydrochloride is a selective, high affinity P2Y12 receptor antagonist that inhibits ADP-induced platelet aggregation. Learn MoreStarting at: $99.00
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ZK 93426 hydrochloride
ZK 93426 hydrochloride is a potent, selective and competitive benzodiazepine receptor antagonist. Learn MoreStarting at: $115.00
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VU 1545
VU 1545 is a metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulator. Learn MoreStarting at: $115.00
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RF 9
RF 9 is a selective NPFF receptor antagonist that blocks NPFF-induced hypothermia and increases in atrial blood pressure and heart rate, and prevents opioid-induced tolerance associated with hyperalgesia in vivo. Learn MoreStarting at: $85.00
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WAY 207024 dihydrochloride
WAY 207024 dihydrochloride is a gonadotropin releasing hormone receptor (GnRH-R) antagonist that exhibits potent affinity with IC50 values of 12 and 71 nM for human and rat GnRH receptors respectively. Learn MoreStarting at: $189.00
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Etonitazenyl isothiocyanate
Etonitazenyl isothiocyanate is an affinity label specific for μ opioid sites. Learn MoreStarting at: $125.00
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FIT
FIT is a selective and irreversible δ-opioid agonist that acts by alkylating the receptor. Learn MoreStarting at: $139.00
