Search results for '1001'

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  • VU 10010

    VU 10010 is a selective allosteric potentiator of M4 acetylcholine receptors that binds to an allosteric site on the receptor increasing affinity for ACh and coupling to G-proteins. Learn More

    Starting at: $129.00

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  • TC-G 1001

    TC-G 1001 is a GPR35 agonist (pEC50 values are 7.59 and 8.36 for β-arrestin and Gαq-i5 Ca2+ assays respectively), which displays 1000-fold greater potency at human GPR35 receptors relative to mouse and rat GPR35 orthologs in an IP1 accumulation assay. Learn More

    Starting at: $139.00

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  • (S)-WAY 100135 dihydrochloride

    (S)-WAY 100135 dihydrochloride is a potent, selective 5-HT1A receptor antagonist (IC50 = 15 nM). Learn More

    Starting at: $110.00

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  • VUF 8430 dihydrobromide

    VUF 8430 dihydrobromide is a high affinity (pKi = 7.5), potent histamine H4 receptor full agonist (pEC50 = 7.3). Displays moderate affinity for H3 receptors (pKi = 6.0) and weak partial agonist activity at H2 receptors. Learn More

    Starting at: $109.00

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4 Item(s)

per page