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XAC
XAC is an adenosine receptor antagonist (IC50 values are 1.8 and 114 nM at A1 and A2 receptors respectively). Learn MoreStarting at: $95.00
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G-1
G-1 is a potent and selective GPR30 receptor agonist that increases cytosolic Ca2+ and inhibits migration of SKBr3 cells and MCF-7 cells in response to chemoattractants with IC50 values of 0.7 and 1.6 nM respectively in vitro. Learn MoreStarting at: $139.00
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ML 221
ML 221 is an apelin receptor (APJ) antagonist with IC50 values of 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively). Learn MoreStarting at: $139.00
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ZK 756326
ZK 756326 is a selective, non-peptide CCR8 chemokine receptor agonist with IC50 values of 1.8 and 2.6 μM for human and mouse receptors respectively. Learn MoreStarting at: $105.00
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Iloprost
Iloprost is a prostacyclin (PGI2) analog that inhibits platelet aggregation induced by collagen, thrombin and ADP with IC50 values of 0.24, 0.71 and 1.07 nM respectively. Learn MoreStarting at: $239.00
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Bucindolol
Bucindolol is a non-selective β-adrenoceptor antagonist with additional α1-adrenoceptor blocking activity. Ki values are 1.61, 1.20 and 68.9 nM for β1-, β2- and α1-adrenoceptors respectively. Learn MoreStarting at: $139.00
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Terazosin hydrochloride
Terazosin hydrochloride is an α1- and α2B-adrenoceptor antagonist with Ki values of 3.3, 0.7, 1.1, 7.7, 1510 and 78.2 nM for α1A, α1B, α1D, α2B, α2A and α2C receptors respectively. Learn MoreStarting at: $70.00
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EMD 386088 hydrochloride
EMD 386088 hydrochloride is a potent 5-HT6 receptor agonist (EC50 = 1.0 nM) that displays selectivity over other 5-HT receptors (IC50 values are 7.4, 110, 180, 240, 450, 620, 660 and 3000 nM for 5-HT6, 5-HT1D, 5-HT1B, 5-HT2A, 5-HT2C, 5-HT4, 5-HT1A and 5-HT7 receptors respectively). Learn MoreStarting at: $99.00
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Conessine
Conessine is a potent and selective histamine H3 receptor antagonist. It is a steroidal alkaloid that displays in vitro antiplasmodial activity (IC50 = 1.04 μM). Learn MoreStarting at: $92.00
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SB 205384
A selective, competitive and orally active GABAB antagonist which displays an IC50 of 1.1 μM at GABAB, approximately 60 times that of CGP 35348 and no binding affinity for GABAA at concentrations up to 100 μM. Learn MoreStarting at: $135.00
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8-Hydroxy-PIPAT oxalate
SCH 58261 is a potent and selective A2A adenosine receptor competitive antagonist (Ki = 1.3 nM). Displays 323-, 53- and 100-fold selectivity over A1, A2B and A3 receptors, respectively. Learn MoreStarting at: $120.00
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L-745,870 trihydrochloride
BIBP 3226 trifluoroacetate is a mixed non-peptide neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor antagonist (Ki values are 1.1, 79, 108, > 1000, > 1000 and >1000 for rNPY Y1, hNPFF2, rNPFF, rNPY Y2, rNPY Y4 and rNPY Y5 respectively). Learn MoreStarting at: $95.00
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Terfenadine
Terfenadine is a histamine H1 receptor antagonist, which also blocks KV11.1 (hERG) and Kir6 (KATP) channels (IC50 values are 204 nM and 1.2 μM respectively). Learn MoreStarting at: $49.00
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HEMADO
HEMADO is an high affinity and selective adenosine A3 receptor agonist (Ki values are 1.1, 327, 1230 and > 30,000 nM for human A3, A1, A2A and A2B receptors respectively). Learn MoreStarting at: $139.00
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MRS 2279
MRS 2279 is a selective, high affinity competitive antagonist of the P2Y1 receptor (Ki = 2.5 nM; IC50 = 51.6 nM). Learn MoreStarting at: $259.00
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2-ThioUTP tetrasodium salt
2-ThioUTP tetrasodium salt is a potent and selective P2Y2 agonist (EC50 values are 0.035, 0.35 and 1.5 μM for hP2Y2, hP2Y4 and hP2Y6 receptors respectively). Learn MoreStarting at: $269.00
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LY 487379 hydrochloride
LY 487379 hydrochloride is a positive allosteric modulator selective for mGlu2 receptors, which potentiates glutamate-stimulated [35S]GTPγS binding (EC50 values are 1.7 and > 10 μM for mGlu2 and mGlu3 receptors respectively). Learn MoreStarting at: $110.00
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TCS 2510
TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM), which displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM. Learn MoreStarting at: $139.00
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LU AA33810
LU AA33810 is a potent neuropeptide Y (NPY) Y5 receptor antagonist (Ki = 1.5 nM in vitro) which displays ≥ 3300-fold affinity for Y5 over Y1, Y2 and Y4 receptors. Learn MoreStarting at: $109.00
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Oleamide
Oleamide endogenous sleep-inducing lipid, which acts as an agonist at the CB1 cannabinoid receptor (EC50 = 1.64 μM). Learn MoreStarting at: $59.00
