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Search results for 'AP 24534'
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GR 89696 fumarate
Highly potent and selective κ-opioid agonist (IC50 = 0.04 nM) that may be selective for the putative κ2 receptor. Learn MoreStarting at: $135.00
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CGP 36216 hydrochloride
CGP 36216 hydrochloride is a selective GABAB antagonist, which displays activity at presynaptic receptors. Learn MoreStarting at: $130.00
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ICI 204,448 hydrochloride
ICI 204,448 hydrochloride is a peripherally acting κ agonist. Learn MoreStarting at: $95.00
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(RS)-PPG
(RS)-PPG is a potent and selective group III metabotropic glutamate receptor agonist, with approximately 25-fold preference for hmGlu8. Learn MoreStarting at: $100.00
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Cyprodime hydrochloride
Cyprodime hydrochloride is a selective μ-opioid receptor antagonist (Ki values are 5.4, 244.6 and 2187 nM for μ-, δ- and κ-opioid receptors respectively). Learn MoreStarting at: $130.00
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Clocinnamox mesylate
Clocinnamox mesylate is a systemically active, irreversible μ-opioid receptor antagonist (apparent Ki values are 0.7, 1.9 and 5.7 nM for mouse μ, δ and κ receptors respectively). Learn MoreStarting at: $95.00
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ICI 199,441 hydrochloride
ICI 199,441 hydrochloride is a highly potent κ agonist, 146-fold more active than U-50488 in vitro. Learn MoreStarting at: $95.00
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U-54494A hydrochloride
U-54494A hydrochloride is a κ-opioid agonist and anticonvulsant, which acts as an NMDA antagonist. Learn MoreStarting at: $105.00
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Naltriben mesylate
Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively), which displays selectivity for the δ2 subtype in vivo. Learn MoreStarting at: $100.00
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Naltrindole hydrochloride
Naltrindole hydrochloride is a highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ and κ opioid receptors. Learn MoreStarting at: $95.00
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Thioperamide
Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist, which blocks eosinophil shape change (IC50 = 1.4 μM) and chemotaxis (IC50 = 519 nM) induced by histamine. Learn MoreStarting at: $90.00
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nor-Binaltorphimine dihydrochloride
nor-Binaltorphimine dihydrochloride is a selective κ-opioid receptor antagonist. Learn MoreStarting at: $90.00
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WEB 2086
WEB 2086 is a potent, selective platelet-activating factor (PAF) receptor antagonist (Ki = 16.3 nM). Which inhibits growth and proliferation of MCF-7 breast cancer cells. Learn MoreStarting at: $75.00
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Z-Cyclopentyl-AP4
Z-Cyclopentyl-AP4 is a group III mGlu receptor agonist that exhibits higher potency at mGlu4 than mGlu8 (EC50 values are 49 and 124 μM respectively) with no activity at mGlu7. And selectively inhibits synaptic activity in the lateral perforant pathway (IC50 values are 130 and 1859 μM in the lateral and medial perforant pathways respectively). Learn MoreStarting at: $129.00
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Devazepide
Devazepide is a potent, orally active CCK1 (CCK-A) receptor antagonist that displays appetite-stimulant effects. Devazepide blocks the anorectic response to CCK-8 and increases food intake in rats following systemic and i.c.v administration. Learn MoreStarting at: $149.00
