Search results for 'AP 24534'

(R)-(-)-α-Methylhistamine dihydrobromide

(R)-(-)-α-Methylhistamine dihydrobromide is a very potent, high affinity H3 agonist that inhibits H3-mediated histamine synthesis and release in the CNS and stimulates H4-mediated eosinophil shape change. Learn More

Starting at: $89.00

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Imetit dihydrobromide

Imetit dihydrobromide is an extremely potent, high affinity agonist at H3 and H4 receptors (Ki values are 0.3 and 2.7 nM respectively), which induces shape change in eosinophils with an EC50 of 25 nM. Learn More

Starting at: $90.00

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Dimaprit dihydrochloride

Dimaprit dihydrochloride is a selective H2 agonist with central effects upon systemic administration, which also inhibits nNOS (IC50 = 49 μM). Learn More

Starting at: $90.00

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Clobenpropit dihydrobromide

Clobenpropit dihydrobromide is an extremely potent histamine H3 antagonist/inverse agonist (pA2=9.93), which displays partial agonist activity at H4 receptors; induces eosinophil shape change with an EC50 of 3 nM. Learn More

Starting at: $115.00

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Thioperamide

Thioperamide is a potent histamine H3 and H4 antagonist/inverse agonist, which blocks eosinophil shape change (IC50 = 1.4 μM) and chemotaxis (IC50 = 519 nM) induced by histamine. Learn More

Starting at: $90.00

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