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Search results for 'inhibit'
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Decynium 22
Decynium 22 is an inhibitor of the plasma membrane monoamine transporter (PMAT) (Ki = 0.10 μM). Learn MoreStarting at: $49.00
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(-)-5'-DMH-CBD
(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable, which displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Learn MoreStarting at: $149.00
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(±)-McN 5652
(±)-McN 5652 is a potent, high affinity serotonin re-uptake inhibitor; selective in viv, and displays moderate selectivity over noradrenalin and dopamine re-uptake in vitro (Ki values are 0.68, 2.9 and 36.8 nM for inhibition of serotonin, noradrenalin and dopamine uptake respectively in rat brain synaptosomes). Learn MoreStarting at: $139.00
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(±)-MDMA hydrochloride
(±)-MDMA hydrochloride is a hallucinogenic compound that inhibits 5-HT and dopamine uptake. Learn MoreStarting at: $105.00
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VU 0240551
VU 0240551 is an inhibitor of the neuronal K-Cl cotransporter, KCC2 that also inhibits hERG and L-type Ca2+ channels. Learn MoreStarting at: $115.00
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Indatraline hydrochloride
Indatraline hydrochloride is a potent monoamine uptake inhibitor that inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET). Learn MoreStarting at: $95.00
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WAY 213613
WAY 213613 is a potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3. Learn MoreStarting at: $139.00
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LY 2365109 hydrochloride
LY 2365109 hydrochloride is a potent and selective glycine transporter 1 (GlyT1) inhibitor that induces a dose-dependent elevation in CSF levels of glycine, and enhances acetylcholine and dopamine release in the striatum and prefrontal cortex respectively. Learn MoreStarting at: $149.00
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YM 244769
YM 244769 is an inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX) that inhibits Na+-dependent 45Ca2+ uptake with IC50 values of 18, 68 and 96 nM for CCL39 cells transfected with NCX3, NCX1 and NCX2 respectively. Learn MoreStarting at: $125.00
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Concanamycin A
Concanamycin A is a specific inhibitor of V-type (vacuolar) H+-ATPase that blocks cell surface expression of virus envelope glycoproteins without affecting synthesis and exhibits cytotoxicity in several cell lines. Learn MoreStarting at: $99.00
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Sertraline hydrochloride
Sertraline hydrochloride is a potent, orally active selective serotonin re-uptake inhibitor (SSRI). Learn MoreStarting at: $109.00
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GBR 13069 dihydrochloride
GBR 13069 dihydrochloride is a potent inhibitor of dopamine uptake with an IC50 value of 40 nM. Learn MoreStarting at: $89.00
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SCH 28080
SCH 28080 is a potent inhibitor of H+,K+-ATPase that binds to the K+ recognition site and is competitive with respect to K+. Learn MoreStarting at: $139.00
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cis-ACBD
cis-ACBD is a potent, competitive and selective inhibitor of glutamate uptake. Learn MoreStarting at: $99.00
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L-(-)-threo-3-Hydroxyaspartic acid
L-(-)-threo-3-Hydroxyaspartic acid is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $149.00
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STF 31
STF 31 is an inhibitor of GLUT1 that inhibits glucose uptake in renal cell carcinoma (RCC) 4 cells. Learn MoreStarting at: $155.00
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Org 24598 lithium salt
Org 24598 lithium salt is a selective inhibitor of the glial glycine transporter (GlyT1). pIC50 values are 6.9, <4 and <3 for GlyT1, GABA transporter and Glyt2 respectively. Learn MoreStarting at: $139.00
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Talopram hydrochloride
Talopram hydrochloride is a potent, selective inhibitor of the noradrenalin transporter (NET) with selectivity for NET against SERT (5-HT transporters) and DAT (dopamine transporters). Learn MoreStarting at: $139.00
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GBR 12783 dihydrochloride
GBR 12783 dihydrochloride is a potent and selective inhibitor of dopamine uptake with IC50 value of 1.8 nM for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes. Learn MoreStarting at: $99.00
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L-trans-2,4-PDC
L-trans-2,4-PDC is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $115.00
