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Search results for 'CT 47098'
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(-)-5'-DMH-CBD
(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable, which displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Learn MoreStarting at: $149.00
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(±)-McN 5652
(±)-McN 5652 is a potent, high affinity serotonin re-uptake inhibitor; selective in viv, and displays moderate selectivity over noradrenalin and dopamine re-uptake in vitro (Ki values are 0.68, 2.9 and 36.8 nM for inhibition of serotonin, noradrenalin and dopamine uptake respectively in rat brain synaptosomes). Learn MoreStarting at: $139.00
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WAY 213613
WAY 213613 is a potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3. Learn MoreStarting at: $139.00
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LY 2365109 hydrochloride
LY 2365109 hydrochloride is a potent and selective glycine transporter 1 (GlyT1) inhibitor that induces a dose-dependent elevation in CSF levels of glycine, and enhances acetylcholine and dopamine release in the striatum and prefrontal cortex respectively. Learn MoreStarting at: $149.00
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BTS 54-505 hydrochloride
BTS 54-505 hydrochloride is a potently active primary amine metabolite of sibutramine. Learn MoreStarting at: $95.00
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YM 244769
YM 244769 is an inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX) that inhibits Na+-dependent 45Ca2+ uptake with IC50 values of 18, 68 and 96 nM for CCL39 cells transfected with NCX3, NCX1 and NCX2 respectively. Learn MoreStarting at: $125.00
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Concanamycin A
Concanamycin A is a specific inhibitor of V-type (vacuolar) H+-ATPase that blocks cell surface expression of virus envelope glycoproteins without affecting synthesis and exhibits cytotoxicity in several cell lines. Learn MoreStarting at: $99.00
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Sertraline hydrochloride
Sertraline hydrochloride is a potent, orally active selective serotonin re-uptake inhibitor (SSRI). Learn MoreStarting at: $109.00
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SCH 28080
SCH 28080 is a potent inhibitor of H+,K+-ATPase that binds to the K+ recognition site and is competitive with respect to K+. Learn MoreStarting at: $139.00
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CGP 37157
CGP 37157 is a selective antagonist of the mitochondrial Na+-Ca2+ exchanger with an IC50 of 0.4 μM. Learn MoreStarting at: $139.00
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cis-ACBD
cis-ACBD is a potent, competitive and selective inhibitor of glutamate uptake. Learn MoreStarting at: $99.00
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Org 24598 lithium salt
Org 24598 lithium salt is a selective inhibitor of the glial glycine transporter (GlyT1). pIC50 values are 6.9, <4 and <3 for GlyT1, GABA transporter and Glyt2 respectively. Learn MoreStarting at: $139.00
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Talopram hydrochloride
Talopram hydrochloride is a potent, selective inhibitor of the noradrenalin transporter (NET) with selectivity for NET against SERT (5-HT transporters) and DAT (dopamine transporters). Learn MoreStarting at: $139.00
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GBR 12783 dihydrochloride
GBR 12783 dihydrochloride is a potent and selective inhibitor of dopamine uptake with IC50 value of 1.8 nM for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes. Learn MoreStarting at: $99.00
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Bicifadine hydrochloride
Bicifadine hydrochloride is an orally active, potent antagonist of the noradrenalin transporter with antagonist activity at the 5-HT and dopamine transporters (IC50 values are 117 nM and 910 nM respectively). Learn MoreStarting at: $139.00
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Paroxetine maleate
Paroxetine maleate is a highly potent and selective 5-HT uptake inhibitor that binds with high affinity to the serotonin transporter. Learn MoreStarting at: $90.00
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(±)-Nipecotic acid
(±)-Nipecotic acid is a GABA uptake inhibitor with IC50 values of 8, 38, 106 and 2370 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively. Learn MoreStarting at: $56.00
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Citalopram hydrobromide
Citalopram hydrobromide is a highly selective and potent 5-HT uptake inhibitor with no effect on noradrenalin or dopamine uptake with IC50 values of 1.8, 8800 and 41000 nM respectively. Learn MoreStarting at: $105.00
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Desipramine hydrochloride
Desipramine hydrochloride is a tricyclic antidepressant that is a selective inhibitor of noradrenalin transporters with Ki values of 4, 61 and 78720 nM for NET, SERT and DAT transporters respectively. Learn MoreStarting at: $41.00
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Paxilline
Paxilline, a potent blocker of high-conductance Ca2+-activated K+ (BKCa, KCa1.1) channels, binds to the α-subunit of BKCa (Ki = 1.9 nM for block of currents in α-subunit-expressing oocytes) and enhances binding of charybdotoxin to BKCa channels in vascular smooth muscle. Learn MoreStarting at: $198.00
