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Search results for 'AG 490'
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Canrenone
Canrenone is a mineralocorticoid receptor antagonist. Learn MoreStarting at: $59.00
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DY131
DY131 is a novel selective agonist at estrogen-related receptors ERRβ and ERRγ that displays minimal activity at ERRα, ERα and ERβ at concentrations up to 30 μM. Learn MoreStarting at: $95.00
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Clofibric acid
Clofibric acid is a PPAR agonist. Learn MoreStarting at: $55.00
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AC 261066
AC 261066 is a potent RARβ2 agonist with a pEC50 value of 8.1. Learn MoreStarting at: $139.00
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Y 134
Y 134 is a selective estrogen receptor modulator (SERM) that acts as an agonist in the bone and antagonist in reproductive tissue. Learn MoreStarting at: $139.00
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UVI 3003
UVI 3003 is a RXR antagonist that displays high RXR binding affinity. Learn MoreStarting at: $115.00
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PHTPP
PHTPP is a selective estrogen ERβ receptor antagonist that exhibits full antagonism at ERβ in a cotransfection assay in human endometrial cancer cells (HEC-1), with minimal effects on ERα. Learn MoreStarting at: $145.00
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RU 28318 (potassium salt)
RU 28318 (potassium salt) is a potent and selective antagonist for the mineralocorticoid receptor (MR) that inhibits aldosterone production and secretion, and selectively decreases ex-vivo MR binding in the hippocampus of adrenalectomised rats. Learn MoreStarting at: $139.00
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RU 26752
RU 26752 is a mineralocorticoid receptor antagonist that prevents aldosterone-induced hypertension in rats. Learn MoreStarting at: $89.00
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SR 202
SR 202 is a selective PPARγ antagonist that inhibits PPARγ-dependent adipocyte differentiation and growth in vitro and in vivo. Learn MoreStarting at: $90.00
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TCPOBOP
TCPOBOP is an agonist of the constitutive androstane receptor that induces activity of ER1 cytochrome P450 isozymes, NADPH-cytochrome c reductase, microsomal epoxide hydrolase and glutathione S transferase. Learn MoreStarting at: $79.00
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Ciglitazone
Ciglitazone is a selective agonist at PPAR&gamma with an EC50 value of 3 μM in vivo. Learn MoreStarting at: $139.00
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Estropipate
Estropipate is an estrogen receptor agonist that inhibits organic anion transporting polypeptide 1B1 (OATP1B1). Learn MoreStarting at: $75.00
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6,2',4'-Trimethoxyflavone
6,2',4'-Trimethoxyflavone is an aryl hydrocarbon receptor antagonist with EC50 value of 0.9 μM. Learn MoreStarting at: $85.00
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CP 775146
CP 775146 is a selective, high affinity PPARα agonist with Ki values of 24.5 nM for PPARα and >10 μM for PPARβ and PPARγ in vitro). Learn MoreStarting at: $169.00
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(Z)-4-Hydroxytamoxifen
(Z)-4-Hydroxytamoxifen is an estrogen receptor antagonist. Learn MoreStarting at: $139.00
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Docosahexaenoic acid
Docosahexaenoic acid is a endogenous omega-3 fatty acid. It acts as a selective retinoid X receptor (RXR) agonist that displays no activity at RAR, thyroid hormone receptor or the vitamin D receptor (VDR). Learn MoreStarting at: $75.00
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AC 55649
AC 55649 is a potent, isoform-selective RARβ2 receptor agonist that displays 100-fold selectivity versus other retinoid receptors. Inhibits proliferation of the breast cancer cell line MCF-7. Learn MoreStarting at: $99.00
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Fexaramine
Fexaramine is a potent, selective farnesoid X receptor agonist with EC50 = 25 nM. Learn MoreStarting at: $155.00
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CD 2665
SC 236 is a selective COX-2 inhibitor (IC50 values are 0.005 and 17.8 μM for COX-2 and COX-1 respectively) which displays anti-inflammatory properties and potent antimetastatic activity against both experimental metastases and spontaneous metastases arising following primary tumor excision. Learn MoreStarting at: $140.00
