Search results for 'inhibitor'

18 Item(s)

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  • ML 298 hydrochloride

    ML 298 hydrochloride is a selective inhibitor of phospholipase D2 (PLD2) (IC50 values are 355 and >20,000 nM for PLD2 and PLD1, respectively), which decreases invasive migration in U87-MG glioblastoma cells, without affecting cell viability. Learn More

    Starting at: $125.00

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  • 9-AC

    9-AC is a Cl- transport inhibitor with a moderate to strong inhibitory action on PKA activated cardiac IcI. Learn More

    Starting at: $65.00

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  • L-Serine

    L-Serine is an endogenous agonist at the inhibitory glycine receptor. Learn More

    Starting at: $33.00

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  • L-Alanine

    L-Alanine is an Agonist at the inhibitory glycine receptor. Learn More

    Starting at: $33.00

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  • T16Ainh-A01

    T16Ainh-A01 is an inhibitor of Ca2+-dependent Cl- channel (CaCC) transmembrane protein 16A (TMEM16A) (IC50 = 1.8 μM in A253 salivary gland epithelial cells). Learn More

    Starting at: $119.00

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  • (-)-[3R,4S]-Chromanol 293B

    680C91 is a potent and selective inhibitor of tryptophan 2,3-dioxygenase (TDO) (Ki = 51 nM) which exhibits no activity against indoleamine 2,3-dioxygenase, monoamine oxidase A and B, 5-HT uptake or 5-HT1A, 1D, 2A and 2C receptors. Learn More

    Starting at: $140.00

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  • ZK 200775

    Benzamil is a Na+/Ca2+ exhanger (NCX) inhibitor (IC50 ~ 100 nM); TRPP3 channel blocker (IC50 = 1.1 μM for inhibition of Ca2+-activated TRPP3 channel activity). Learn More

    Starting at: $140.00

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  • DMP 543

    Indirubin-3'-oxime is aprotein kinase inhibitor and inhibits cyclin-dependent kinases (IC50 = 0.18 - 3.33 μM) and GSK-3β (IC50 = 0.19 μM). Learn More

    Starting at: $95.00

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  • Vinpocetine

    Vinpocetine is a phosphodiesterase inhibitor, selective for PDE1 (IC50 = 21 μM), which also blocks voltage-gated Na+ channels. Learn More

    Starting at: $109.00

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  • CaCCinh-A01

    Calcium-activated chloride channel (CaCC) inhibitor (IC50 ~ 10 μM), which inhibits CaCC currents in human bronchial and intestinal cells. Learn More

    Starting at: $99.00

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  • NS 3623

    NS 3623 is a human ether-a-go-go (hERG) KV11.1 potassium channel activator, which activates the IKr current and displays antiarrhythmic activity and exhibits potential dual mode of action at the hERG inhibitory site; may also act as a partial blocker of KV11.1 (hERG) channels. Learn More

    Starting at: $145.00

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  • Hypotaurine

    Endogenous inhibitory amino acid. Learn More

    Starting at: $75.00

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  • Arcaine sulfate

    Arcaine sulfate is a NO synthase inhibitor, acting as a competitive inhibitor at the polyamine site. Learn More

    Starting at: $80.00

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  • ML 218 hydrochloride

    ML 218 hydrochloride is a selective inhibitor of T-type calcium channels (IC50 values are 270 and 310 nM for Cav3.3 and Cav3.2 respectively in a patch EP assay). Learn More

    Starting at: $169.00

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  • SKF 96365 hydrochloride

    SKF 96365 hydrochloride is a store-operated Ca2+ entry (SOCE) inhibitor that inhibits STIM1.It also blocks TRPC channels, voltage-gated Ca2+ channels and potassium channels. Learn More

    Starting at: $115.00

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  • Phenamil

    Phenamil is TRPP3 channel inhibitor (IC50 = 0.14 μM), which also inhibits epithelial Na+ channels (Kd = 0.4 nM for a high affinity site on the epithelial Na+ channel). Learn More

    Starting at: $55.00

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  • EIPA

    EIPA is a TRPP3 channel inhibitor (IC50 = 10.5 μM), which inhibits the Na+/H+ exchanger (NHE). Learn More

    Starting at: $65.00

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  • β-Alanine

    β-Alanine is a non-specific endogenous agonist at the inhibitory glycine receptor. More selective than taurine, which slso distinguishes between GABA transporters (IC50 values are 19, 58, 110, 1320 and 5690 μM for rGAT-2, hGAT-3, rGAT-3, hBGT-3 and hGAT-1 respectively). Learn More

    Starting at: $49.00

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18 Item(s)

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