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Search results for 'PI'
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(R)-(+)-Bay K 8644
(R)-(+)-Bay K 8644 is a L-type Ca2+-channel blocker with negative inotropic and vasodilatatory effects in vivo. Learn MoreStarting at: $189.00
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(S)-(-)-Bay K 8644
(S)-(-)-Bay K 8644 is a L-type Ca2+-channel activator with positive inotropic, vasoconstrictive and behavioral effects in vivo. Learn MoreStarting at: $199.00
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Levcromakalim
Levcromakalim is an active enantiomer of the prototypical Kir6 (KATP) channel opener cromakalim. Learn MoreStarting at: $169.00
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Cromakalim
Cromakalim is a prototypical Kir6 (KATP) channel opener that relaxes rabbit isolated portal vein with an IC50 value of 21 nM . Learn MoreStarting at: $139.00
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Benidipine hydrochloride
Benidipine hydrochloride is an orally active antihypertensive agent that inhibits L-, N- and T-type Ca2+ channels and also inhibits aldosterone-induced mineralocorticoid receptor activation. Learn MoreStarting at: $109.00
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TC-P 262
TC-P 262 is a selective P2X3 and P2X2/3 receptor antagonist (pIC50 values are 7.39 and 6.68 respectively). Learn MoreStarting at: $109.00
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6-Iodonordihydrocapsaicin
6-Iodonordihydrocapsaicin is a potent competitive vanilloid TRPV1 (VR1) receptor antagonist that inhibits capsaicin-induced [Ca2+]i increase in rat DRG neurons, and guinea pig bladder and trachea contractions in vitro. Learn MoreStarting at: $115.00
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Mirtazapine
Mirtazapine is an antidepressant agent that enhances noradrenalin (NA) release in rat brain via inhibition of α2-adrenergic autoreceptors and displays only weak affinity for monoamine transporters. Learn MoreStarting at: $85.00
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(±)-LY 395756
(±)-LY 395756, an analog of LY 354740, is a selective metabotropic glutamate ligand for mGlu2 and mGlu3 receptors. Learn MoreStarting at: $199.00
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DCPIB
DCPIB is a potent, selective blocker of the volume-sensitive anion channel (VSAC) that reverses cell swelling-induced action potential duration shortening in atrial myocytes and inhibits astroglial swelling in vitro. Learn MoreStarting at: $109.00
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4-Acetyl-1,1-dimethylpiperazinium iodide
4-Acetyl-1,1-dimethylpiperazinium iodide is a structural analog of acetylcholine that acts as a nicotinic agonist with a Ki value of 29.9 nM at α4β2. Learn MoreStarting at: $89.00
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Amperozide hydrochloride
Amperozide hydrochloride is a typical antipsychotic that displays high affinity for 5-HT2 receptors and low affinity for D2 receptors. Learn MoreStarting at: $99.00
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Piracetam
Piracetam is a nootropic that displays cognitive enhancing properties.It facilitates efficiency of cholinergic neurotransmission at muscarinic receptors. Learn MoreStarting at: $55.00
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(RS)-AMPA
(RS)-AMPA is a prototypical and defining agonist for the AMPA subgroup of ionotropic glutamate receptors. Learn MoreStarting at: $139.00
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1-Acetyl-4-methylpiperazine hydrochloride
1-Acetyl-4-methylpiperazine hydrochloride is a structural analog of acetylcholine that acts as a nAChR agonist. Learn MoreStarting at: $96.00
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DCEBIO
DCEBIO stimulates Cl- secretion via the activation of hKCa3.1 (IK1) potassium channels and an apical Cl- conductance carried by the CFTR channel. Learn MoreStarting at: $99.00
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TCN 213
TCN 213 is a NMDA receptor antagonist, selective for NR1/NR2A (pIC50 = 5.4) over NR1/NR2B. Learn MoreStarting at: $149.00
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T16Ainh-A01
T16Ainh-A01 is an inhibitor of Ca2+-dependent Cl- channel (CaCC) transmembrane protein 16A (TMEM16A) (IC50 = 1.8 μM in A253 salivary gland epithelial cells). Learn MoreStarting at: $119.00
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MRS 1845
MRS 1845 is potent blocker of store-operated Ca2+ channels and inhibits capacitative Ca2+ influx in HL-60 cells (IC50 = 1.7 mM). Learn MoreStarting at: $120.00
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L-Quisqualic acid
L-Quisqualic acid is a glutamate receptor agonist acting at AMPA receptors and metabotropic glutamate receptors positively linked to phosphoinositide hydrolysis. Learn MoreStarting at: $65.00
