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Search results for 'LY 215840'
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ML 298 hydrochloride
ML 298 hydrochloride is a selective inhibitor of phospholipase D2 (PLD2) (IC50 values are 355 and >20,000 nM for PLD2 and PLD1, respectively), which decreases invasive migration in U87-MG glioblastoma cells, without affecting cell viability. Learn MoreStarting at: $125.00
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L-651,582
L-651,582 is an orally active Ca2+ channel blocker which inhibits K+- and carbachol-stimulated Ca2+ influx (IC50 values are 500 and 935 nM respectively). Learn MoreStarting at: $149.00
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RN 1734
RN 1734 is a selective TRPV4 antagonist with IC50 values of 2.3, 5.9 and 3.2 μM for hTRPV4, mTRPV4 and rTRPV4 receptors respectively. Learn MoreStarting at: $95.00
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Benidipine hydrochloride
Benidipine hydrochloride is an orally active antihypertensive agent that inhibits L-, N- and T-type Ca2+ channels and also inhibits aldosterone-induced mineralocorticoid receptor activation. Learn MoreStarting at: $109.00
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LY 2087101
LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs. Learn MoreStarting at: $125.00
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Cl-HIBO
Cl-HIBO is a subtype-selective and strongly desensitising AMPA receptor agonist. Learn MoreStarting at: $179.00
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Zacopride hydrochloride
Zacopride hydrochloride is a highly potent 5-HT3 receptor antagonist and 5-HT4 receptor agonist with Ki values of 0.38nM and 373nM respectively. Learn MoreStarting at: $105.00
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HC 067047
HC 067047 is a potent and selective TRPV4 antagonist that reversibly inhibits currents through mouse, human and rat TRPV4 orthologs. Learn MoreStarting at: $139.00
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TC-P 262
TC-P 262 is a selective P2X3 and P2X2/3 receptor antagonist (pIC50 values are 7.39 and 6.68 respectively). Learn MoreStarting at: $109.00
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A 844606
A 844606 is a selective α7 nicotinic acetylcholine receptor (nAChR) agonist with EC50 values of 1.4 and 2.2 μM at human and rat receptors respectively. Learn MoreStarting at: $129.00
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Mirtazapine
Mirtazapine is an antidepressant agent that enhances noradrenalin (NA) release in rat brain via inhibition of α2-adrenergic autoreceptors and displays only weak affinity for monoamine transporters. Learn MoreStarting at: $85.00
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(±)-LY 395756
(±)-LY 395756, an analog of LY 354740, is a selective metabotropic glutamate ligand for mGlu2 and mGlu3 receptors. Learn MoreStarting at: $199.00
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MG 624
MG 624 inhibits α-Bgtx binding to chick α7 and α4β2 subtypes with Ki values of 106 nM and 84 μM respectively. Learn MoreStarting at: $99.00
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(RS)-4-Carboxyphenylglycine
(RS)-4-Carboxyphenylglycine is a broad spectrum EAA ligand. Learn MoreStarting at: $99.00
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Psora 4
Psora 4 is a potent KV1.3 channel blocker (EC50 = 3 nM) that preferentially binds the C-type inactivated state of the channel. Learn MoreStarting at: $145.00
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NS 3763
NS 3763 is a selective non-competitive kainate receptor antagonist that displays selectivity for GLUK5 subunit-containing receptors with IC50 values of 1.6 and > 30 μM for homomeric GLUK5 and GLUK6 receptors respectively. Learn MoreStarting at: $99.00
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TCN 237 dihydrochloride
TCN 237 dihydrochloride is a highly potent NR2B-selective NMDA receptor antagonist that blocks NR2B-mediated calcium influx in Ltk cells with Ki value of 9.7 nM). Learn MoreStarting at: $115.00
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Chlorisondamine diiodide
Chlorisondamine diiodide is an exceptionally long lasting nicotinic antagonist with IC50 value of ~1.6 mM. Learn MoreStarting at: $99.00
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PPDA
PPDA is a subtype-selective NMDA receptor antagonist that preferentially binds to NR2C/NR2D-containing receptors. Learn MoreStarting at: $119.00
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Nonactin
Nonactin is a monovalent cation ionophore that displays selectivity for K+ and NH4+. It also inhibits P-glycoprotein-mediated efflux of chemotherapeutic agents in multiple-drug resistant cancer cells. Learn MoreStarting at: $99.00
