You have no items in your shopping cart.
Search results for 'AP 24534'
-
6-Iodonordihydrocapsaicin
6-Iodonordihydrocapsaicin is a potent competitive vanilloid TRPV1 (VR1) receptor antagonist that inhibits capsaicin-induced [Ca2+]i increase in rat DRG neurons, and guinea pig bladder and trachea contractions in vitro. Learn MoreStarting at: $115.00
-
Mirtazapine
Mirtazapine is an antidepressant agent that enhances noradrenalin (NA) release in rat brain via inhibition of α2-adrenergic autoreceptors and displays only weak affinity for monoamine transporters. Learn MoreStarting at: $85.00
-
RuBi-4AP
RuBi-4AP is a water soluble ruthenium-bipyridine-triphenylphosphine caged 4-aminopyridine (4-AP). Learn MoreStarting at: $119.00
-
A 784168
A 784168 is a potent TRPV1 antagonist with an IC50 value of 25 nM for inhibition of TRPV1 activation by 50 nM capsaicin. Learn MoreStarting at: $139.00
-
JNJ 17203212
JNJ 17203212 is a reversible, competitive and potent TRPV1 antagonist that inhibits capsaicin- and H+-induced channel activation and exhibits antitussive and analgesic activity in vivo. Learn MoreStarting at: $119.00
-
D-AP7
D-AP7 is a more active form of AP7. Learn MoreStarting at: $179.00
-
D-AP5
D-AP5 is a competitive NMDA antagonist. Learn MoreStarting at: $59.00
-
L-AP5
L-AP5 is a NMDA antagonist and also an agonist at quisqualate-sensitized AP6 site. Learn MoreStarting at: $145.00
-
DL-AP7
DL-AP7 is a phosphono NMDA antagonist. Learn MoreStarting at: $79.00
-
L-AP6
L-AP6 is a selective agonist for 'quis'-sensitized site. Learn MoreStarting at: $179.00
-
D-AP4
D-AP4 is a broad spectrum excitatory amino acid receptor antagonist. Learn MoreStarting at: $169.00
-
Cesium chloride
Cesium chloride is a potassium channel blocker that prevents activation of caspase-3 and neuronal apoptosis in serum- and potassium-deprived cerebellar granule neurons by inactivating GSK-3β. Learn MoreStarting at: $39.00
-
DL-AP5
DL-AP5 is a potent NMDA antagonist. Learn MoreStarting at: $65.00
-
Nonactin
Nonactin is a monovalent cation ionophore that displays selectivity for K+ and NH4+. It also inhibits P-glycoprotein-mediated efflux of chemotherapeutic agents in multiple-drug resistant cancer cells. Learn MoreStarting at: $99.00
-
(±)-Anatoxin A fumarate
(±)-Anatoxin A fumarate is a potent nicotinic agonist that stimulates [3H]-dopamine release from rat striatal synaptosomes with EC50 value of 136 nM. Learn MoreStarting at: $139.00
-
DCEBIO
DCEBIO stimulates Cl- secretion via the activation of hKCa3.1 (IK1) potassium channels and an apical Cl- conductance carried by the CFTR channel. Learn MoreStarting at: $99.00
-
AP 18
AP 18 is a Reversible TRPA1 channel blocker with IC50 values of 3.1 and 4.5 μM at human and mouse TRPA1 respectively. Learn MoreStarting at: $90.00
-
MRS 1845
MRS 1845 is potent blocker of store-operated Ca2+ channels and inhibits capacitative Ca2+ influx in HL-60 cells (IC50 = 1.7 mM). Learn MoreStarting at: $120.00
-
2-APB
2-APB is a functional and membrane permeable D-myo-inositol 1,4,5-trisphosphate (IP3) receptor antagonist with IC50 = 42 μM. Learn MoreStarting at: $45.00
-
DMP 543
Indirubin-3'-oxime is aprotein kinase inhibitor and inhibits cyclin-dependent kinases (IC50 = 0.18 - 3.33 μM) and GSK-3β (IC50 = 0.19 μM). Learn MoreStarting at: $95.00
