Bromodomains
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UNC 1215
UNC 1215 is a potent inhibitor of L3MBTL3 methyllysine (Kme) reader domain (IC50 = 40 nM; Kd = 120 nM), which displays >100-fold selectivity over a panel of histone methyltransferases, kinases, ion channels and 7-TM receptors. Learn MoreStarting at: $149.00
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Galloflavin
Galloflavin is an inhibitor of human lactate dehydrogenase (LDH) (Ki values are 5.46 and 15.1 μM for LDH-A and LDH-B, respectively, in competition with pyruvate), which inhibits lactate production and decreases ATP synthesis in PLD/PRF/5 cells. Learn MoreStarting at: $109.00
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GPP 78 hydrochloride
GPP 78 hydrochloride is an inhibitor of nicotinamide phosphoribosyltransferase (NMPRTase); potently depletes NAD levels and exhibits cytotoxicity in vitro (IC50 values are 3.0 and 3.8 nM respectively). Learn MoreStarting at: $169.00