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Peptide Receptors
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SB 657510
SB 657510 is a selective urotensin-II (UT) receptor antagonist (Ki values are 61, 17, 30, 65 and 56 nM at human, monkey, cat, rat and mouse receptors respectively), which inhibits U-II-induced intracellular Ca2+ mobilization (IC50 = 180 nM) and antagonizes the contractile action of U-II in isolated mammalian arteries and aortae (EC50 = 50 - 189 nM). Learn MoreStarting at: $139.00
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(±)-AC 7954 hydrochloride
(±)-AC 7954 hydrochloride is a highly selective, non-peptide urotensin-II (UT) receptor agonist that displays potent activity at human and rat UT receptors (pEC50 values are 6.5 and 6.7 respectively). Learn MoreStarting at: $139.00
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SB 706375
SB 706375 is a high affinity, non-peptide antagonist of the urotensin-II (UT) receptor with high affinity for mammalian UT receptors, including human, mouse and rat (Ki values are 9.3, 19.1 and 20.7 nM respectively, in HEK293 cells expressing recombinant UT receptors). Learn MoreStarting at: $139.00
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OPC 21268
OPC 21268 is a nonpeptide vasopressin V1 receptor antagonist, which displays greater affinity for rat V1 than human V1 (Ki values are 25 and 8800 nM respectively). Learn MoreStarting at: $150.00
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SR 49059
SR 49059 is a potent and selective non-peptide vasopressin V1A receptor antagonist; devoid of agonist activity, which displays high affinity and efficacy at both rat (Ki = 1.6 nM) and human (Ki = 1.1 - 6.3 nM) V1A receptors. Learn MoreStarting at: $225.00
