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Nicotinic (α7) Receptors
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AR-R 17779 hydrochloride
AR-R 17779 hydrochloride is a selective agonist of α7 nAChRs (Ki values are 190 and 16000 nM for rat α7 and α4β2 receptors respectively). Learn MoreStarting at: $140.00
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LY 2087101
LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs. Learn MoreStarting at: $125.00
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SEN 12333
SEN 12333 is a α7 nicotinic acetylcholine receptor (nAChR) agonist that displays functional antagonism at histamine H3 receptors (IC50 = 103 nM) and weak agonist activity at human ganglionic α3 nAChRs with an IC50 value of 8.5 μM. Learn MoreStarting at: $125.00
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A 844606
A 844606 is a selective α7 nicotinic acetylcholine receptor (nAChR) agonist with EC50 values of 1.4 and 2.2 μM at human and rat receptors respectively. Learn MoreStarting at: $129.00
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MG 624
MG 624 inhibits α-Bgtx binding to chick α7 and α4β2 subtypes with Ki values of 106 nM and 84 μM respectively. Learn MoreStarting at: $99.00
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TC 1698 dihydrochloride
TC 1698 dihydrochloride is a selective nicotinic α7 receptor agonist that displays weak partial agonist/antagonist activity at β-subunit-containing receptors. Learn MoreStarting at: $125.00
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PHA 568487
PHA 568487 is an orally active and brain penetrant agonist of the α7 nicotinic acetylcholine receptor (Ki values are 44 and 2800 for α7 and 5-HT3 respectively). Learn MoreStarting at: $99.00
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NS 1738
NS 1738 is a selective positive allosteric modulator of α7 nicotinic acetylcholine receptors. Exhibits no substantial activity for α4β2, α3β3 and α1-containing receptors. Learn MoreStarting at: $99.00
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PHA 543613 hydrochloride
PHA 543613 hydrochloride is a potent α7 nAChR agonist that displays selectivity over α3β4, α1β1γδ, α4β2 and 5-HT3 receptors, which positively influences sensory gating and memory in in vivo models of schizophrenia. Learn MoreStarting at: $149.00
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TQS
TQS is a type II positive allosteric modulator of α7 nACh receptors (pEC50 = 5.5). Learn MoreStarting at: $125.00
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DMAB-anabaseine dihydrochloride
DMAB-anabaseine dihydrochloride is a partial agonist at α7-containing neuronal nicotinic receptors and antagonist at α4β2 and other nicotinic receptors. Learn MoreStarting at: $119.00
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S 24795
S 24795 is a partial agonist of α7 nAChR, which improves mnemonic function in aged mice for the treatment of aging-related memory disturbances and displays more efficient memory-enhancing effects than memantine in Alzheimer's disease mouse models. Learn MoreStarting at: $90.00
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CCMI
CCMI is a positive allosteric modulator of α7 neuronal nicotinic acetylcholine receptors (nAChR) that evokes positive modulation of acetylcholine (ACh)-induced EC5 currents. Learn MoreStarting at: $95.00
