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Neurotransmitter Transporters
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3-CPMT
3-CPMT binds with high affinity to the dopamine transporter (Ki = 30 nM) and blocks re-uptake of dopamine. Learn MoreStarting at: $50.00
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Threo-methylphenidate hydrochloride
Psychomotor stimulant. Inhibitor of dopamine and noradrenalin transporters that increases the extracellular concentration of dopamine and noradrenalin. Learn MoreStarting at: $85.00
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Mephedrone hydrochloride
Mephedrone hydrochloride Inhibits striatal dopamine uptake and hippocampal 5-HT uptake in synaptosomes (IC50 values are 467 and 558 nM respectively). Learn MoreStarting at: $95.00
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Bupropion hydrochloride
Bupropion hydrochloride is a non-selective inhibitor of dopamine and noradrenalin transporters (Ki values are 1.4, 2.8 and 45 μM for NET, DAT and SERT transporters respectively), which also inhibits neuronal nicotinic acetylcholine receptors. Learn MoreStarting at: $99.00
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3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride is a potent inhibitor of dopamine uptake and transport (Ki = 11.8 nM). Learn MoreStarting at: $75.00
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TFB-TBOA
TFB-TBOA is a high affinity, selective blocker of glial glutamate transporters EAAT1 and EAAT2 (IC50 values are 17, 22 and 300 nM for EAAT2, EAAT1 and EAAT3 respectively), which displays no activity on a wide range of neurotransmitter receptors and transporters. Learn MoreStarting at: $89.00
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L-(-)-threo-3-Hydroxyaspartic acid
L-(-)-threo-3-Hydroxyaspartic acid is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $149.00
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cis-ACBD
cis-ACBD is a potent, competitive and selective inhibitor of glutamate uptake. Learn MoreStarting at: $99.00
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7-Chlorokynurenic acid sodium salt
7-Chlorokynurenic acid sodium salt is a sodium salt of 7-Chlorokynurenic acid, an NMDA receptor antagonist acting at the glycine site. Learn MoreStarting at: $65.00
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L-trans-2,4-PDC
L-trans-2,4-PDC is a potent, competitive, transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor. Learn MoreStarting at: $115.00
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WAY 213613
WAY 213613 is a potent, non-substrate inhibitor of EAAT2 (GLT-1) that displays > 44-fold selectivity over EAAT1 and EAAT3. Learn MoreStarting at: $139.00
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L-CCG-lll
L-CCG-lll is a potent and competitive inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate. Learn MoreStarting at: $265.00
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7-Chlorokynurenic acid
7-Chlorokynurenic acid is a NMDA receptor antagonist acting at the glycine site. Potent competitive inhibitor of L-glutamate transport into synaptic vesicles. Learn MoreStarting at: $60.00
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Ceftriaxone disodium salt
Ceftriaxone disodium salt is β-lactam antibiotic, which increased activity of the EAAT2 glutamate transporter and displays neuroprotective activity in vivo via upregulation. Learn MoreStarting at: $49.00
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MPDC
MM 77 dihydrochloride is a highly potent and fairly selective 5-HT1A ligand, which may be a full antagonist at postsynaptic receptors. Learn MoreStarting at: $135.00
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Dihydrokainic acid
Dihydrokainic acid is a EAAT2(GLT1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake. Learn MoreStarting at: $49.00
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Evans Blue tetrasodium salt
Evans Blue tetrasodium salt is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits AMPA and kainate receptor-mediated currents (IC50 values are 220 and 150 nM respectively). Learn MoreStarting at: $65.00
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(±)-HIP-B
(±)-HIP-B is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.2 μM) rather than [3H]L-glutamate uptake (IC50 = 16.9 μM). Learn MoreStarting at: $139.00
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(±)-HIP-A
(±)-HIP-A is a potent, non-competitive excitatory amino acid transporter (EAAT) blocker which preferentially inhibits glutamate-induced [3H]D-aspartate release (IC50 = 1.6 μM) rather than [3H]L-glutamate uptake (IC50 = 18 μM). Learn MoreStarting at: $139.00
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DL-TBOA
DL-TBOA is a competitive, non-transportable blocker of excitatory amino acid transporters (IC50 values are 70, 6, and 6 μM for EAAT1, EAAT2 and EAAT3 respectively), which also inhibits EAAT4 and EAAT5 (Ki values are 4.4 and 3.2 μM respectively). Learn MoreStarting at: $140.00
