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Ligand-gated Ion Channels
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Quinolinic acid
Quinolinic acid is an endogenous NMDA agonist and transmitter candidate. Learn MoreStarting at: $59.00
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SEN 12333
SEN 12333 is a α7 nicotinic acetylcholine receptor (nAChR) agonist that displays functional antagonism at histamine H3 receptors (IC50 = 103 nM) and weak agonist activity at human ganglionic α3 nAChRs with an IC50 value of 8.5 μM. Learn MoreStarting at: $125.00
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A 844606
A 844606 is a selective α7 nicotinic acetylcholine receptor (nAChR) agonist with EC50 values of 1.4 and 2.2 μM at human and rat receptors respectively. Learn MoreStarting at: $129.00
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MNI-caged-D-aspartate
MNI-caged-D-aspartate is a D-aspartate caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $149.00
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CGS 19755
CGS 19755 is a potent, competitive NMDA receptor antagonist. Learn MoreStarting at: $129.00
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DL-AP5
DL-AP5 is a potent NMDA antagonist. Learn MoreStarting at: $65.00
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QNZ 46
QNZ 46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist (IC50 values are 3, 6, 229, and >300, >300 μM for NR2D, NR2C, NR2A, NR2B, and GluR1, respectively). Learn MoreStarting at: $130.00
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PPDA
PPDA is a subtype-selective NMDA receptor antagonist that preferentially binds to NR2C/NR2D-containing receptors. Learn MoreStarting at: $119.00
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(R)-CPP
(R)-CPP is a highly potent NMDA antagonist, which shows some selectivity for NR2A-containing receptors (Ki values are 0.041, 0.27, 0.63 and 1.99 μM for inhibition of NR2A-, NR2B-, NR2C- and NR2D-containing recombinant NMDA receptors respectively). Learn MoreStarting at: $245.00
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LY 233053
LY 233053 is a competitive NMDA receptor antagonist (IC50 = 7 nM) that displays no affinity for AMPA or kainate receptors at a concentration of 10 μM, and nhibits NMDA-induced neuronal degeneration and protects from NMDA-induced convulsions in neonatal rats. Learn MoreStarting at: $65.00
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(R)-(+)-HA-966
(R)-(+)-HA-966 is an antagonist/partial agonist at the glycine site of the NMDA receptor. Learn MoreStarting at: $95.00
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MNI-caged-NMDA
MNI-caged-NMDA is a NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $175.00
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TC 1698 dihydrochloride
TC 1698 dihydrochloride is a selective nicotinic α7 receptor agonist that displays weak partial agonist/antagonist activity at β-subunit-containing receptors. Learn MoreStarting at: $125.00
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TCN 237 dihydrochloride
TCN 237 dihydrochloride is a highly potent NR2B-selective NMDA receptor antagonist that blocks NR2B-mediated calcium influx in Ltk cells with Ki value of 9.7 nM). Learn MoreStarting at: $115.00
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threo Ifenprodil hemitartrate
threo Ifenprodil hemitartrate is a potent σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist. Learn MoreStarting at: $109.00
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Dextromethorphan hydrobromide
Dextromethorphan hydrobromide is a Non-competitive, low affinity NMDA receptor antagonist with the effect of antitussive, anticonvulsive and neuroprotective. Learn MoreStarting at: $42.00
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(S)-(-)-HA-966
(S)-(-)-HA-966 is a possesses potent sedative and ataxic action, probably through disruption of striatal dopaminergic mechanisms. Learn MoreStarting at: $95.00
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D-CPP-ene
D-CPP-ene is a potent and competitive NMDA antagonist (Ki = 40 nM). Learn MoreStarting at: $270.00
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Eliprodil
Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site. Learn MoreStarting at: $90.00
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CGP 37849
CGP 37849 is a potent, selective and competitive NMDA receptor antagonist (Ki = 35 nM). Learn MoreStarting at: $115.00
