Glutamate (Metabotropic) Receptors
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CHIR 99021 trihydrochloride
CHIR 99021 trihydrochloride is a hydrochloride salt of CHIR 99021, a highly selective GSK-3 inhibitor. Learn MoreStarting at: $189.00
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EGLU
EGLU is a selective antagonist of presynaptically-mediated (1S,3S)-ACPD-induced depression of motoneuron excitation in neonatal rat spinal cord; presumed group II mGlu receptor antagonist. Learn MoreStarting at: $110.00
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Xanthurenic acid
Xanthurenic acid attenuates cAMP formation in mouse cortical slices expressing mGlu2 and mGlu3 receptors. Learn MoreStarting at: $39.00
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MAP4
(S)-SNAP 5114 is a GABA transport inhibitor, showing selectivity for GAT-3 and GAT-2 (IC50 values are 5, 21 and 388 μM for hGAT-3, rGAT-2 and hGAT-1 respectively). Learn MoreStarting at: $135.00
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MTPG
RS 17053 hydrochloride is a α1A-adrenoceptor antagonist, with very high affinity for α1A receptors (pKi and pA2 estimates of 9.1 - 9.9) and a 30 - 100 fold selectivity over the α1B and α1D subtypes (pKi and pA2 estimates 7.7 - 7.8). Learn MoreStarting at: $135.00
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DCG IV
DCG IV is a presynaptic depressant; highly potent agonist for group II mGlu receptors. Learn MoreStarting at: $135.00
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ACPT-II
ACPT-II is a competitive metabotropic receptor antagonist (KB values are 115, 88 and 77 μM at mGlu1a, mGlu2 and mGlu4a respectively). Learn MoreStarting at: $140.00
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L-Glutamic acid
L-Glutamic is the predominant excitatory transmitter in the mammalian central nervous system. It acts at ionotropic and metabotropic glutamate receptors. Learn MoreStarting at: $32.00