GABA Receptors
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THIP hydrochloride
THIP hydrochloride is a systemically active GABAA receptor agonist and GABAC receptor antagonist with antinociceptive, anticonvulsant and sedative effects. Learn MoreStarting at: $109.00
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CL 218872
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors. Learn MoreStarting at: $60.00
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Lorazepam
Lorazepam is a ligand at the GABAA receptor benzodiazepine modulatory site. Learn MoreStarting at: $75.00
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PK 11195
PK 11195 possesses high affinity for the MDR (peripheral benzodiazepine receptor) without binding to other known neurotransmitter receptors. Learn MoreStarting at: $69.00
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ZK 93426 hydrochloride
ZK 93426 hydrochloride is a potent, selective and competitive benzodiazepine receptor antagonist. Learn MoreStarting at: $115.00
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Ro 15-4513
Ro 15-4513 is a high affinity benzodiazepine ligand that acts as partial inverse agonist at recombinant DS α1-, α2-, α3- and α5-GABAA receptors. Learn MoreStarting at: $115.00
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ZAPA sulfate
ZAPA sulfate is a useful ligand to investigate GABA receptors linked to benzodiazepine receptors. It is also a GABAC receptor antagonist. Learn MoreStarting at: $95.00
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DPNI-Caged GABA
DPNI-Caged GABA is a nitroindoline-caged GABA with similar photochemical properties to MNI-glutamate. Learn MoreStarting at: $335.00
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AA 29504
AA 29504 is a positive allosteric modulator of GABAA receptors that modulates both α4β3δ-containing extrasynaptic receptors and α1β3γ2S-containing receptors in Xenopus oocytes. Learn MoreStarting at: $139.00
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Ocinaplon
Ocinaplon is a modulator of GABAA receptors, which displays modest selectivity for GABAA α1 receptors; and partial agonist activity at α2-, α3- and α5-containing receptors. Learn MoreStarting at: $139.00
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β-CCB
β-CCB is an endogenous proconvulsant and anxiogenic benzodiazepine receptor ligand. Learn MoreStarting at: $79.00
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ZK 93423 hydrochloride
ZK 93423 hydrochloride is a potent benzodiazepine receptor agonist. Learn MoreStarting at: $129.00
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(R)-Baclofen
(R)-Baclofen is a selective GABAB agonist. Learn MoreStarting at: $59.00
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17-PA
17-PA is a selective antagonist of neurosteroid potentiation and direct gating of GABAA receptors. Learn MoreStarting at: $159.00
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3-Methyl-GABA
3-Methyl-GABA is an activator of GABA aminotransferase. Learn MoreStarting at: $90.00
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(-)-Bicuculline methobromide
(-)-Bicuculline methobromide is a methobromide salt of (+)-bicuculline. Learn MoreStarting at: $85.00
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MRK 016
MRK 016 is a GABAA receptor inverse agonist selective for the α5-subtype that exhibits affinity at benzodiazepine binding site of recombinant human GABAA receptors. Learn MoreStarting at: $149.00
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FG 7142
FG 7142 is an inverse agonist and anxiogenic agent that increases tyrosine hydroxylation and causes upregulation of β-adrenoceptors in mouse cerebral cortex. Learn MoreStarting at: $119.00
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Dihydroergotoxine mesylate
Dihydroergotoxine mesylate binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. Learn MoreStarting at: $79.00
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Zolpidem
Zolpidem is a benzodiazepine agonist with high selectivity for α1-subunit-containing GABAA receptors (BZ/ω1 site) and very high intrinsic activity. Learn MoreStarting at: $119.00