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Dopamine Receptors
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PNU 177864 hydrochloride
PNU 177864 hydrochloride is a highly selective dopamine D3 receptor antagonist which induces phospholipidosis and exhibits antischizophrenic activity in vivo. Learn MoreStarting at: $109.00
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PG 01037 dihydrochloride
PG 01037 dihydrochloride is a Dopamine D3 receptor antagonist with 133-fold selectivity for D3 over D2 receptors in vitro (Ki values are 0.70, 93.3 and 375 nM for D3, D2 and D4 receptors respectively). Learn MoreStarting at: $139.00
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NGB 2904
NGB 2904 is a potent and selective dopamine D3 receptor antagonist (Ki values are 1.4, 217, 223, 642, > 5000, > 10000 and > 10000 nM for D3, D2, 5-HT2, α1, D4, D1 and D5 receptors respectively). Learn MoreStarting at: $135.00
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GSK 789472 hydrochloride
GSK 789472 hydrochloride is a selective dopamine D3 receptor antagonist and D2 partial agonist (pEC50 values are <5.5 and 8.3 respectively), which selective against the D4 receptor in both agonist and antagonist assays. Brain penetrant. Learn MoreStarting at: $95.00
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U 99194 maleate
U 99194 maleateis a potent, selective D3 antagonist. Learn MoreStarting at: $109.00
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Nafadotride
Nafadotride is a highly potent, competitive, preferential dopamine D3 receptor antagonist. Ki values are 0.52, 5, and 269 nM for human cloned D3, D2 and D4 receptors respectively. Learn MoreStarting at: $135.00
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ABT 724 trihydrochloride
ABT 724 trihydrochloride is a potent dopamine D4 receptor partial agonist. Learn MoreStarting at: $109.00
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L-745,870 trihydrochloride
BIBP 3226 trifluoroacetate is a mixed non-peptide neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor antagonist (Ki values are 1.1, 79, 108, > 1000, > 1000 and >1000 for rNPY Y1, hNPFF2, rNPFF, rNPY Y2, rNPY Y4 and rNPY Y5 respectively). Learn MoreStarting at: $95.00
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L-741,742 hydrochloride
L-741,742 hydrochloride is a potent and highly selective D4 dopamine receptor antagonist, with Ki values of > 1700, 770 and 3.5 nM at cloned human D2, D3 and D4 receptors. Learn MoreStarting at: $95.00
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PD 168077 maleate
PD 168077 maleate is a potent D4 dopamine receptor agonist (Ki = 8.7 nM) that induces synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons. Learn MoreStarting at: $119.00
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Ro 10-5824 dihydrochloride
Ro 10-5824 dihydrochloride is a selective dopamine D4 receptor partial agonist (EC50 = 205 nM) that binds with high affinity (Ki = 5.2 nM). Learn MoreStarting at: $98.00
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Sonepiprazole
Sonepiprazole is a selective, high affinity antagonist for the rat and human dopamine D4 receptor (Ki = 10 nM). Learn MoreStarting at: $140.00
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PNU 96415E
PNU 96415E is antipsychotic agent which displays high affinity for dopamine D4 and serotonergic 5-HT2A receptors and relatively weak affinity at D2 receptors (Ki values are 3.0, 5.8, 134, 181, 199, 240, 411 and > 678 nM for D4, 5-HT2A, 5-HT1A, α1, D2, D3, D1, α2 and muscarinic receptors respectively). Learn MoreStarting at: $95.00
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NGD 94-1
NGD 94-1 is a high affinity D4 receptor ligand; selective over D1, D2, D3 and D5 receptors. Displays antagonist activity at the human D4.2 receptor (Ki = 3.6 nM in transfected CHO cells) and exhibits agonist activity at the D4.4 receptor in HEK 293 cells. Learn MoreStarting at: $110.00
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PD 168568 dihydrochloride
PD 168568 dihydrochloride is a potent and selective dopamine D4 receptor antagonist (Ki values are 8.8 and 1842 nM at D4 and D2 receptors respectively). Learn MoreStarting at: $105.00
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A 412997 dihydrochloride
A 412997 dihydrochloride is a selective agonist for the dopamine D4 receptor (Ki values are 7.9 and 12.1 nM for human D4 and rat D4 receptors) which shows efficacy in rat models of ADHD and short-term memory. Learn MoreStarting at: $95.00
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Raclopride
Raclopride is a selective and potent dopamine D2/D3 receptor antagonist. Learn MoreStarting at: $69.00
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(-)-Quinpirole hydrochloride
(-)-Quinpirole hydrochloride is a selective dopamine D2 receptor agonist. Learn MoreStarting at: $95.00
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NPEC-caged-dopamine
NPEC ((N)-1-(2-nitrophenyl)ethyl) caged version of dopamine which releases dopamine leading to D1 receptor activation upon UV light illumination (360 nm), and Induces PKA activation and c-Fos expression in cortical and striatal neurons, with striatal neurons demonstrating a significantly greater detection and sensitivity to sub-second dopamine signals as compared to cortical neurons. Learn MoreStarting at: $120.00
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(+)-AJ 76 hydrochloride
(+)-AJ 76 hydrochloride is a dopamine receptor antagonist with preferential action at presynaptic receptors. Learn MoreStarting at: $115.00
