μ Opioid Receptors
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Clocinnamox mesylate
Clocinnamox mesylate is a systemically active, irreversible μ-opioid receptor antagonist (apparent Ki values are 0.7, 1.9 and 5.7 nM for mouse μ, δ and κ receptors respectively). Learn MoreStarting at: $95.00
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Cyprodime hydrochloride
Cyprodime hydrochloride is a selective μ-opioid receptor antagonist (Ki values are 5.4, 244.6 and 2187 nM for μ-, δ- and κ-opioid receptors respectively). Learn MoreStarting at: $130.00
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Oxycodone hydrochloride
Oxycodone hydrochloride is a potent and selective μ-opioid receptor agonist (Ki values are 16 and >1000 nM for hMOR1 and hKOR1 respectively). Learn MoreStarting at: $65.00
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β-Funaltrexamine hydrochloride
β-Funaltrexamine hydrochloride is a selective μ opioid receptor antagonist. Learn MoreStarting at: $149.00
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Naloxonazine dihydrochloride
Naloxonazine dihydrochloride is a potent opioid antagonist, selective for μ1 receptors. Learn MoreStarting at: $79.00
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Etonitazenyl isothiocyanate
Etonitazenyl isothiocyanate is an affinity label specific for μ opioid sites. Learn MoreStarting at: $125.00
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Fentanyl citrate
Fentanyl citrate is a potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively), which displays antinociceptive activity in vivo. Learn MoreStarting at: $55.00