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Search results for 'AP 24534'
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NPEC-caged-D-AP5
NPEC-caged-D-AP5 is a D-AP5 caged with the photosensitive 1-(2-nitrophenyl)ethoxycarbonyl (NPEC) group. NMDA receptor antagonist. Learn MoreStarting at: $189.00
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Fentanyl citrate
Fentanyl citrate is a potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively), which displays antinociceptive activity in vivo. Learn MoreStarting at: $55.00
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Ocinaplon
Ocinaplon is a modulator of GABAA receptors, which displays modest selectivity for GABAA α1 receptors; and partial agonist activity at α2-, α3- and α5-containing receptors. Learn MoreStarting at: $139.00
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(+)-UH 232 maleate
(+)-UH 232 maleate is a D2 antagonist (Ki = 72.7 nM in a ligand binding assay; apparent KB = 14.5 nM in a cAMP accumulation assay), which displays preferential activity at central dopamine autoreceptors. Learn MoreStarting at: $109.00
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Ipsapirone
Ipsapirone is a selective 5-HT1A receptor agonist with a Ki value of 10 nM. Learn MoreStarting at: $99.00
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AA 29504
AA 29504 is a positive allosteric modulator of GABAA receptors that modulates both α4β3δ-containing extrasynaptic receptors and α1β3γ2S-containing receptors in Xenopus oocytes. Learn MoreStarting at: $139.00
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ZAPA sulfate
ZAPA sulfate is a useful ligand to investigate GABA receptors linked to benzodiazepine receptors. It is also a GABAC receptor antagonist. Learn MoreStarting at: $95.00
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W146
W146 is a potent sphingosine-1-phosphate receptor S1P1 selective antagonist that enhances capillary leakage and restores lymphocyte egress in vivo. Learn MoreStarting at: $109.00
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ML 221
ML 221 is an apelin receptor (APJ) antagonist with IC50 values of 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively). Learn MoreStarting at: $139.00
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Trap 101
Trap 101 is a potent and selective nociceptin/orphanin FQ (NOP) receptor antagonist. Learn MoreStarting at: $139.00
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(+)-AJ 76 hydrochloride
(+)-AJ 76 hydrochloride is a dopamine receptor antagonist with preferential action at presynaptic receptors. Learn MoreStarting at: $115.00
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Salvinorin A
Salvinorin A displays high affinity at both native (Ki = 4.3 nM) and cloned (Ki = 16 nM) κ-opioid receptors. Learn MoreStarting at: $139.00
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(R)-(-)-α-Methylhistamine dihydrobromide
(R)-(-)-α-Methylhistamine dihydrobromide is a very potent, high affinity H3 agonist that inhibits H3-mediated histamine synthesis and release in the CNS and stimulates H4-mediated eosinophil shape change. Learn MoreStarting at: $89.00
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Nemonapride
Nemonapride is a highly potent dopamine D2-like receptor antagonist. Learn MoreStarting at: $139.00
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(±)-U-50488 hydrochloride
(±)-U-50488 hydrochloride is as elective κ-opioid agonist. Learn MoreStarting at: $99.00
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MSOP
MSOP is a selective group III metabotropic glutamate receptor antagonist that displays an apparent KDof 51 μM for the L-AP4-sensitive presynaptic mGluR on primary afferent terminals in spinal cord compared to > 700 μM for the (1S,3S)-ACPD-sensitive presynaptic mGlu in the same system. Learn MoreStarting at: $138.00
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Urapidil hydrochloride
Urapidil hydrochloride is an α1-adrenoceptor antagonist and 5-HT1A receptor agonist. Learn MoreStarting at: $99.00
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PD 168077 maleate
PD 168077 maleate is a potent D4 dopamine receptor agonist (Ki = 8.7 nM) that induces synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons. Learn MoreStarting at: $119.00
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McN-A 343
McN-A 343 is a selective muscarinic M1 receptor agonist with selectivity for M1 over other muscarinic receptor types appears to arise from a high efficacy at M1 receptors. Learn MoreStarting at: $37.00
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Isamoltane hemifumarate
Isamoltane hemifumarate is a 5-HT1B antagonist, approximately 30-fold selective over 5-HT1A. Learn MoreStarting at: $89.00
