Search results for 'AP 24534'

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  • (±)-McN 5652

    (±)-McN 5652 is a potent, high affinity serotonin re-uptake inhibitor; selective in viv, and displays moderate selectivity over noradrenalin and dopamine re-uptake in vitro (Ki values are 0.68, 2.9 and 36.8 nM for inhibition of serotonin, noradrenalin and dopamine uptake respectively in rat brain synaptosomes). Learn More

    Starting at: $139.00

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  • GBR 12783 dihydrochloride

    GBR 12783 dihydrochloride is a potent and selective inhibitor of dopamine uptake with IC50 value of 1.8 nM for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes. Learn More

    Starting at: $99.00

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  • MPDC

    MM 77 dihydrochloride is a highly potent and fairly selective 5-HT1A ligand, which may be a full antagonist at postsynaptic receptors. Learn More

    Starting at: $135.00

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  • (S)-SNAP 5114

    BTS is a selective inhibitor of the ATPase activity of skeletal muscle myosin II subfragment 1 (S1) (IC50 ~ 5 mM), reversibly blocks gliding motility and suppresses force and twitch production in fast skeletal muscle. Learn More

    Starting at: $135.00

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  • Evans Blue tetrasodium salt

    Evans Blue tetrasodium salt is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits AMPA and kainate receptor-mediated currents (IC50 values are 220 and 150 nM respectively). Learn More

    Starting at: $65.00

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  • Ochratoxin A

    Ochratoxin A is a mycotoxin that increases activity of the endoplasmic reticulum ATP-dependent calcium pump which induces JNK activation and apoptosis in MDCK-C7 cells at nanomolar concentrations. Learn More

    Starting at: $69.00

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  • 7-Chlorokynurenic acid

    7-Chlorokynurenic acid is a NMDA receptor antagonist acting at the glycine site. Potent competitive inhibitor of L-glutamate transport into synaptic vesicles. Learn More

    Starting at: $60.00

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  • (S)-Duloxetine hydrochloride

    (S)-Duloxetine hydrochloride is a high affinity, competitive 5-HT and noradrenaline (NA) re-uptake inhibitor (Ki values are 8.5 and 45 nM for 5-HTand NA reuptake respectively in cortical synaptosomes, which exhibits antidepressant and anxiolytic effects. Learn More

    Starting at: $45.00

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  • Mephedrone hydrochloride

    Mephedrone hydrochloride Inhibits striatal dopamine uptake and hippocampal 5-HT uptake in synaptosomes (IC50 values are 467 and 558 nM respectively). Learn More

    Starting at: $95.00

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  • Chicago Sky Blue 6B

    Chicago Sky Blue 6B is a potent inhibitor of L-glutamate uptake into synaptic vesicles, which inhibits macrophage migration inhibitory factor (MIF) (IC50 = 0.81 μM) and MIF proinflammatory activity. Learn More

    Starting at: $49.00

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