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Search results for 'Anandamide'
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(-)-5'-DMH-CBD
(-)-5'-DMH-CBD is an anandamide membrane transport inhibitor (IC50 = 14 μM) that is relatively metabolically stable, which displays some affinity for CB2 receptors but has only weak affinity for CB1 receptors and has no activity at VR1 receptors or FAAH. Learn MoreStarting at: $149.00
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Anandamide - d4
Anandamide - d4 is a deuterated anandamide that is used as an internal standard for the quantification of AEA by GC- or LC-mass spectrometry. Learn MoreStarting at: $149.00
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Anandamide
Anandamide is an endogenous cannabinoid and TRPV1 receptor agonist that also blocks TNF-α-induced NF-κB activation via direct inhibition of IKK. Learn MoreStarting at: $59.00
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OMDM-2
OMDM-2 is a metabolically stable inhibitor of anandamide cellular uptake that displays relatively low affinity for CB1 and CB2 receptors with Ki values of 5.1 and > 10 μM and for vanilloid VR1 receptors with EC50 value of 10 μM. Learn MoreStarting at: $65.00
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Olvanil
Olvanil, a potent vanilloid receptor agonist, blocks anandamide uptake (IC50 = 9 μM) and may bind to CB1 cannabinoid receptors. Learn MoreStarting at: $99.00
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O-1918
O-1918 is a selective, silent antagonist of a putative endothelial anandamide receptor distinct from CB1 or CB2 receptors. Learn MoreStarting at: $149.00
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O-2093
O-2093 is an inhibitor of anandamide uptake (IC50 = 17.3 μM) with little or no activity at CB1, CB2, TRPV1 and FAAH. Learn MoreStarting at: $99.00
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UCM 707
UCM 707 is a potent endocannabinoid transport inhibitor. IC50 values are 0.8 and 30 μM for inhibition of the anandamide transporter and FAAH respectively. Ki values are 4700, 67 and > 5000 nM for CB1, CB2 and VR1 receptors respectively. Learn MoreStarting at: $125.00
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VDM 11
VDM 11 is a potent and selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4-11 μM, which displays negligible agonist activity at the hVR1 receptor and very weak action at CB1 and CB2 receptors. Learn MoreStarting at: $75.00
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Virodhamine
Virodhamine endogenous cannabinoid receptor mixed agonist/antagonist found in higher concentrations peripherally than anandamide. Learn MoreStarting at: $79.00
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AM 1172
AM 1172 metabolically stable anandamide uptake inhibitor (IC50 = 2.1 - 2.5 μM) and fatty acid amide hydrolase (FAAH) inhibitor (Ki = 3.18 μM). Learn MoreStarting at: $139.00
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AM 404
AM 404 is a competitive and selective inhibitor of carrier-mediated anandamide transport (IC50 = 1 μM). Does not activate CB1 receptors or inhibit anandamide hydrolysis but has been shown to activate native and cloned vanilloid receptors (pEC50 = 7.4). Active in vivo. Also available in water soluble emulsion . Learn MoreStarting at: $65.00
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Palmitoylisopropylamide
Palmitoylisopropylamide is an inhibitor of fatty acid amide hydrolase (FAAH); pIC50 = 4.89 for inhibition of [3H]-anandamide metabolism. Learn MoreStarting at: $65.00
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MAFP
MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). It also binds irreversibly to CB1 receptors (IC50 = 20 nM). Learn MoreStarting at: $98.00
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N-Arachidonylglycine
N-Arachidonylglycine is an endogenous anandamide-like compound. Learn MoreStarting at: $85.00
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(R)-(+)-Methanandamide
(R)-(+)-Methanandamide is a stable anandamide analog that is a selective agonist for the CB1 receptor (Ki values are 20 and 815 nM for CB1 and CB2 receptors respectively), which also displays agonist activity at vanilloid receptors. Learn MoreStarting at: $65.00
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DEA
DEA is a potent endocannabinoid and anandamide analog that activates CB1 receptors in microglia and binds to rat synaptosomal membranes (Ki = 34.4 nM). Learn MoreStarting at: $80.00
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AACOCF3
AACOCF3 is an inhibitor of cytosolic (85 kDa) phospholipase A2. It also inhibits fatty acid amide hydrolase (FAAH, anandamide amidase) in vitro. Learn MoreStarting at: $65.00
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PALDA
PALDA is an endogenous fatty acid dopamide that displays 'entourage' effects on endovanilloids NADA and anandamide. Learn MoreStarting at: $75.00
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Arvanil
Arvanil is a cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist (Ki values are 0.5 and 0.3 μM respectively), which also inhibits the anandamide transporter (IC50 = 3.6 μM). Learn MoreStarting at: $50.00
