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Cannabinoid Receptors
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Bay 59-3074
Bay 59-3074 is a novel CB1/CB2 receptor partial agonist (Ki values are 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively). Learn MoreStarting at: $139.00
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Virodhamine
Virodhamine endogenous cannabinoid receptor mixed agonist/antagonist found in higher concentrations peripherally than anandamide. Learn MoreStarting at: $79.00
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Cannabigerol
Cannabigerol is a partial agonist of CB2 and CB1 receptors (Ki values are 337 and 440 nM respectively) which also exhibits α2-adrenoceptor agonist activity (EC50 = 0.2 nM in mouse brain membranes). Learn MoreStarting at: $155.00
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(-)-Cannabidiol
(-)-Cannabidiol is a non-psychotropic constituent of cannabis that is anticonvulsive, antihyperalgesic and neuroprotective in vivo. Learn MoreStarting at: $110.00
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WIN 55,212-3 mesylate
WIN 55,212-3 mesylate is a novel, low potency CB2 receptor silent antagonist and CB1 receptor partial inverse agonist, which competitively antagonizes effects of CP 55,940 (pA2 = 6.1) and SR 144528 (pEC50 = 5.3) at CB2 receptors and acts as a partial inverse agonist at CB1 receptors (pIC50 = 5.5). Learn MoreStarting at: $90.00
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HU 210
HU 210 is a highly potent cannabinoid receptor agonist (Ki values are 0.061 and 0.52 nM at cloned human CB1 and CB2 receptors respectively), which also displays agonist activity at GPR55 (EC50 = 26 nM). Learn MoreStarting at: $120.00
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2-Palmitoylglycerol
2-Palmitoylglycerol is an endogenous fatty acid glycerol ester that enhances activity of 2-arachidonylglycerol. Learn MoreStarting at: $55.00
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Palmitoylisopropylamide
Palmitoylisopropylamide is an inhibitor of fatty acid amide hydrolase (FAAH); pIC50 = 4.89 for inhibition of [3H]-anandamide metabolism. Learn MoreStarting at: $65.00
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MAFP
MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). It also binds irreversibly to CB1 receptors (IC50 = 20 nM). Learn MoreStarting at: $98.00
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Arachidonyl serotonin
Arachidonyl serotonin is a dual fatty acid amide hydrolase (FAAH) inhibitor/TRPV1 antagonist (IC50 values are 5.6 μM and 37 - 40 nM for FAAH and TRPV1 respectively). Learn MoreStarting at: $75.00
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N-Arachidonylglycine
N-Arachidonylglycine is an endogenous anandamide-like compound. Learn MoreStarting at: $85.00
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O-1918
O-1918 is a selective, silent antagonist of a putative endothelial anandamide receptor distinct from CB1 or CB2 receptors. Learn MoreStarting at: $149.00
