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Cannabinoid Receptors
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AM 630
Immepip dihydrobromide is a potent histamine H3 receptor agonist which also binds to H4 receptors (Ki values are 0.4 and 9 nM at human recombinant H3 and H4 receptors respectively). Learn MoreStarting at: $135.00
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GP 1a
GP 1a is a highly selective CB2 receptor agonist that increases P-ERK1/2 expression in HL-60 cells in vitro with Ki values are 0.037 and 363 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $150.00
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CB 65
CB 65 is a high affinity and selective CB2 receptor agonist. Learn MoreStarting at: $139.00
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GP 2a
GP 2a is a selective CB2 receptor agonist with Ki values of 7.6 and 900 nM for CB2 and CB1 receptors respectively. Learn MoreStarting at: $169.00
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L-759,656
Highly selective CB2 receptor agonist (Ki values are 11.8 and 4888 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 3.1 nM). Learn MoreStarting at: $180.00
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SER 601
SER 601 is a potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Learn MoreStarting at: $109.00
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L-759,633
L-759,633 is a high affinity, selective CB2 receptor agonist (Ki values are 6.4 and 1043 nM for CB2 and CB1 receptors respectively) which potently inhibits forskolin-stimulated cAMP production via CB2 receptors expressed in CHO cells (EC50 = 8.1 nM). Learn MoreStarting at: $180.00
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GW 405833
GW 405833 is a potent and selective CB2 receptor partial agonist (EC50 = 0.65 nM; maximum inhibition = 44.6%) which binds with high affinity to both human and rat CB2 receptors and displays ~ 1200-fold selectivity over CB1 (Ki values are 3.92 and 4772 nM for human recombinant CB2 and CB1 receptors respectively). Learn MoreStarting at: $135.00
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JWH 015
JWH 015 is a selective CB2 agonist (Ki values are 13.8 and 383 nM as measured at human cloned CB2 and CB1 receptors expressed in CHO cells). Learn MoreStarting at: $50.00
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O-1602
O-1602 is an analog of cannabidiol that is a potent agonist at the GPR55 cannabinoid receptor (EC50 values are 13, > 30000 and > 30000 nM for GPR55, CB1 and CB2 receptors respectively). Learn MoreStarting at: $145.00
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Abn-CBD
Neurobehaviorally inactive cannabinoid that acts as a selective agonist for GPR55 (EC50 values are 2.5, >30 and >30 μM at GPR55, CB1 and CB2 receptors respectively). Learn MoreStarting at: $179.00
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CID 16020046
CID 16020046 is a selective GPR55 antagonist that inhibits LPI-induced Ca2+ signaling with an IC50 value of 0.21 μM in HEK-GPR55 cells. Learn MoreStarting at: $139.00
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Oleylethanolamide
Oleylethanolamide is a lipid mediator and analog of anandamide that is involved in peripheral regulation of feeding, which induces satiety through activation of PPARα and is also a ceramidase inhibitor. Learn MoreStarting at: $60.00
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Palmitoylethanolamide
Palmitoylethanolamide, a selective GPR55 agonist, is a substrate for fatty acid amide hydrolase (FAAH) and PEA-preferring acid amidase (PAA) and exhibits antinociceptive and anticonvulsant in vivo. Learn MoreStarting at: $65.00
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WIN 55,212-3 mesylate
WIN 55,212-3 mesylate is a novel, low potency CB2 receptor silent antagonist and CB1 receptor partial inverse agonist, which competitively antagonizes effects of CP 55,940 (pA2 = 6.1) and SR 144528 (pEC50 = 5.3) at CB2 receptors and acts as a partial inverse agonist at CB1 receptors (pIC50 = 5.5). Learn MoreStarting at: $90.00
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2-Arachidonylglycerol
2-Arachidonylglycerol is a endogenous cannabinoid ligand that acts as a potent agonist at GPR55 (EC50 values are 3, 519 and 618 nM at GPR55, CB1 and CB2 respectively; Ki values are 472 and 1400 nM at CB1 and CB2 respectively). Learn MoreStarting at: $132.00
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CP 55940
CP 55940 is a cannabinoid agonist that displays high and roughly equal affinity for both central and peripheral cannabinoid receptors. Learn MoreStarting at: $189.00
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O-2545 hydrochloride
O-2545 hydrochloride is a high affinity, water-soluble CB1/CB2 receptor agonist. Learn MoreStarting at: $105.00
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Cannabinol
Cannabinol, a CB2 and CB1 receptor agonist, inhibits adenylyl cyclase (EC50 values are 120 and 261 nM for CB1 and CB2 receptors respectively) and suppresses immune cell function. Learn MoreStarting at: $149.00
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(-)-Cannabidiol
(-)-Cannabidiol is a non-psychotropic constituent of cannabis that is anticonvulsive, antihyperalgesic and neuroprotective in vivo. Learn MoreStarting at: $110.00
