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Cannabinoid Receptors
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N-Arachidonylglycine
N-Arachidonylglycine is an endogenous anandamide-like compound. Learn MoreStarting at: $85.00
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O-1918
O-1918 is a selective, silent antagonist of a putative endothelial anandamide receptor distinct from CB1 or CB2 receptors. Learn MoreStarting at: $149.00
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Arachidonyl serotonin
Arachidonyl serotonin is a dual fatty acid amide hydrolase (FAAH) inhibitor/TRPV1 antagonist (IC50 values are 5.6 μM and 37 - 40 nM for FAAH and TRPV1 respectively). Learn MoreStarting at: $75.00
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MAFP
MAFP is a potent, irreversible inhibitor of fatty acid amide hydrolase (FAAH, anandamide amidase), the enzyme responsible for anandamide hydrolysis (IC50 = 2.5 nM). It also binds irreversibly to CB1 receptors (IC50 = 20 nM). Learn MoreStarting at: $98.00
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Palmitoylisopropylamide
Palmitoylisopropylamide is an inhibitor of fatty acid amide hydrolase (FAAH); pIC50 = 4.89 for inhibition of [3H]-anandamide metabolism. Learn MoreStarting at: $65.00
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2-Palmitoylglycerol
2-Palmitoylglycerol is an endogenous fatty acid glycerol ester that enhances activity of 2-arachidonylglycerol. Learn MoreStarting at: $55.00
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Bay 59-3074
Bay 59-3074 is a novel CB1/CB2 receptor partial agonist (Ki values are 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively). Learn MoreStarting at: $139.00
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CB 13
CB 13 is a potent, orally active CB1/CB2 receptor agonist with limited brain penetration (EC50 values are 6.1 and 27.9 nM for CB1 and CB2 receptors respectively), which displays antihyperalgesic activity in a rat model of neuropathic pain with no CNS side effects. Learn MoreStarting at: $95.00
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Cannabinol
Cannabinol, a CB2 and CB1 receptor agonist, inhibits adenylyl cyclase (EC50 values are 120 and 261 nM for CB1 and CB2 receptors respectively) and suppresses immune cell function. Learn MoreStarting at: $149.00
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(-)-Cannabidiol
(-)-Cannabidiol is a non-psychotropic constituent of cannabis that is anticonvulsive, antihyperalgesic and neuroprotective in vivo. Learn MoreStarting at: $110.00
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Virodhamine
Virodhamine endogenous cannabinoid receptor mixed agonist/antagonist found in higher concentrations peripherally than anandamide. Learn MoreStarting at: $79.00
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2-Arachidonylglycerol
2-Arachidonylglycerol is a endogenous cannabinoid ligand that acts as a potent agonist at GPR55 (EC50 values are 3, 519 and 618 nM at GPR55, CB1 and CB2 respectively; Ki values are 472 and 1400 nM at CB1 and CB2 respectively). Learn MoreStarting at: $132.00
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Anandamide - d4
Anandamide - d4 is a deuterated anandamide that is used as an internal standard for the quantification of AEA by GC- or LC-mass spectrometry. Learn MoreStarting at: $149.00
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HU 210
HU 210 is a highly potent cannabinoid receptor agonist (Ki values are 0.061 and 0.52 nM at cloned human CB1 and CB2 receptors respectively), which also displays agonist activity at GPR55 (EC50 = 26 nM). Learn MoreStarting at: $120.00
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WIN 55,212-3 mesylate
WIN 55,212-3 mesylate is a novel, low potency CB2 receptor silent antagonist and CB1 receptor partial inverse agonist, which competitively antagonizes effects of CP 55,940 (pA2 = 6.1) and SR 144528 (pEC50 = 5.3) at CB2 receptors and acts as a partial inverse agonist at CB1 receptors (pIC50 = 5.5). Learn MoreStarting at: $90.00
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Cannabigerol
Cannabigerol is a partial agonist of CB2 and CB1 receptors (Ki values are 337 and 440 nM respectively) which also exhibits α2-adrenoceptor agonist activity (EC50 = 0.2 nM in mouse brain membranes). Learn MoreStarting at: $155.00
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O-2545 hydrochloride
O-2545 hydrochloride is a high affinity, water-soluble CB1/CB2 receptor agonist. Learn MoreStarting at: $105.00
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CP 55940
CP 55940 is a cannabinoid agonist that displays high and roughly equal affinity for both central and peripheral cannabinoid receptors. Learn MoreStarting at: $189.00
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Oleylethanolamide
Oleylethanolamide is a lipid mediator and analog of anandamide that is involved in peripheral regulation of feeding, which induces satiety through activation of PPARα and is also a ceramidase inhibitor. Learn MoreStarting at: $60.00
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CID 16020046
CID 16020046 is a selective GPR55 antagonist that inhibits LPI-induced Ca2+ signaling with an IC50 value of 0.21 μM in HEK-GPR55 cells. Learn MoreStarting at: $139.00
