7-TM Receptors

Items 61 to 80 of 819 total

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  • Tocrifluor T1117

    Tocrifluor T1117 is a novel fluorescent form of AM 251, which conjugated with 5-carboxytetramethylrhodamine (5-TAMRA) that fluoresces at 543nm excitation (590nm emission), and displays GPR55 binding activity. Learn More

    Starting at: $200.00

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  • VU 0255035

    VU 0255035 is a highly selective muscarinic M1 antagonist (Ki = 14.87 nM), which targets the M1 orthosteric site and reduces pilocarpine-induced seizures in mice. Learn More

    Starting at: $110.00

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  • CY 208-243

    CY 208-243 is a centrally active dopamine D1 receptor agonist, selective over D2 receptor sites, which stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM, that exerts antiParkinsonian activity in animal models. Learn More

    Starting at: $139.00

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  • DPCPX

    DPCPX is a potent and selective A1 adenosine receptor antagonist, both in vitro and in vivo. Learn More

    Starting at: $119.00

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  • Z-Cyclopentyl-AP4

    Z-Cyclopentyl-AP4 is a group III mGlu receptor agonist that exhibits higher potency at mGlu4 than mGlu8 (EC50 values are 49 and 124 μM respectively) with no activity at mGlu7. And selectively inhibits synaptic activity in the lateral perforant pathway (IC50 values are 130 and 1859 μM in the lateral and medial perforant pathways respectively). Learn More

    Starting at: $129.00

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  • (±)-5'-Chloro-5'-deoxy-ENBA

    (±)-5'-Chloro-5'-deoxy-ENBA is a highly selective adenosine A1 receptor agonist (Ki values are 0.51, 1290, 1340 and 2740 nM at A1, A3, A2A and A2B receptors respectively). Learn More

    Starting at: $135.00

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  • SKF 77434 hydrobromide

    SKF 77434 hydrobromide is a selective dopamine D1-like receptor partial agonist (IC50 values are 19.7 and 2425 nM for binding to D1-like and D2-like receptors respectively). Learn More

    Starting at: $79.00

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  • Cevimeline hydrochloride

    Cevimeline hydrochloride is a selective M1 receptor agonist which induces atropine-sensitive contractions of isolated guinea pig ilea and trachea preparations (EC50 values are 3.5 and 3 μM respectively). Learn More

    Starting at: $95.00

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  • VU 0155041

    VU 0155041 is a potent, positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50 = 798 and 693 nM at human and rat mGlu4 receptors respectively). Learn More

    Starting at: $120.00

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  • Naltrindole hydrochloride

    Naltrindole hydrochloride is a highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ and κ opioid receptors. Learn More

    Starting at: $95.00

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  • Naltriben mesylate

    Naltriben mesylate is a selective and potent δ-opioid receptor antagonist (Ki values are 0.013, 19 and 152 nM for δ, μ and κ receptors respectively), which displays selectivity for the δ2 subtype in vivo. Learn More

    Starting at: $100.00

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  • VU 0357017 hydrochloride

    VU 0357017 hydrochloride is a positive allosteric modulator of muscarinic M1 receptors (EC50 = 198 nM), which displays no activity at M2-M5 at concentrations up to 30 μM. Learn More

    Starting at: $110.00

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  • A 68930 hydrochloride

    A 68930 hydrochloride is a potent and selective D1-like dopamine receptor agonist (EC50 values are 2.1 and 3910 nM for D1-like and D2-like receptors respectively). Learn More

    Starting at: $115.00

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  • SDZ WAG 994

    SDZ WAG 994 is a potent and selective A1 adenosine receptor agonist (Ki values are 23, > 10000 and 25000 nM for A1, A2A and A2B receptors respectively). Learn More

    Starting at: $145.00

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  • SNC 162

    SNC 162 is a potent and selective non-peptide δ-opioid receptor agonist (Ki = 0.63 nM) which displays > 8000-fold selectivity over μ-opioid receptors and is centrally active following systemic administration in vivo. Learn More

    Starting at: $160.00

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  • CPPG

    CPPG is a potent group II/III mGlu receptor antagonist, with approximately 20-fold selectivity for group III over group II (IC50 values of 2.2 and 46.2 nM respectively). Learn More

    Starting at: $115.00

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  • ACPT-I

    ACPT-I is an agonist for group III mGlu receptors (EC50 values are 7.2 and 8.2 μM for mGlu4a and mGlu8 respectively). Learn More

    Starting at: $140.00

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  • HTMT dimaleate

    HTMT dimaleate is a H1 and H2 receptor agonist, which increases intracellular Ca2+ and IP3 in lymphocytes through a binding site other than H1, H2 or H3. And 4x104 times more active than histamine in H2-mediated effects in natural suppressor cells. Learn More

    Starting at: $98.00

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  • NADA

    NADA is a potent endogenous cannabinoid and vanilloid receptor agonist, with no action at dopamine receptors. Selective for CB1 over CB2 receptors (Ki values are 0.25 and 12 μM respectively), and potent agonist at TRPV1 (VR1) receptors (EC50 ~ 50 nM). Learn More

    Starting at: $79.00

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  • (S)-3,4-DCPG

    (S)-3,4-DCPG is a potent, selective mGlu8a agonist (EC50 = 31 nM). Displays > 100-fold selectivity over mGlu1-7, which increases c-Fos expression in stress-related brain areas following systemic administration in mice in vivo. Learn More

    Starting at: $140.00

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