You have no items in your shopping cart.
7-TM Receptors
-
VU 0364770
VU 0364770 is a positive allosteric modulator at mGlu4 receptors with EC50 of 290 nM in mGlu4-expressing HEK 293 cells that prevents attentional deficit and forelimb asymmetry in a rodent model of Parkinson's disease. Learn MoreStarting at: $109.00
-
Oxprenolol hydrochloride
Oxprenolol hydrochloride is a non-selective β-adrenergic antagonist. Learn MoreStarting at: $59.00
-
TC-C 14G
TC-C 14G is a potent, high affinity CB1 receptor inverse agonist with high efficacy in a hypothermia assay (ID50 = 5 mg/kg) in vivo. Learn MoreStarting at: $140.00
-
MSOP
MSOP is a selective group III metabotropic glutamate receptor antagonist that displays an apparent KDof 51 μM for the L-AP4-sensitive presynaptic mGluR on primary afferent terminals in spinal cord compared to > 700 μM for the (1S,3S)-ACPD-sensitive presynaptic mGlu in the same system. Learn MoreStarting at: $138.00
-
Fenoldopam hydrochloride
Fenoldopam hydrochloride is a selective D1-like dopamine receptor partial agonist with EC50 value of 57 nM. Learn MoreStarting at: $119.00
-
(±)-CP 47497
(±)-CP 47497 is a potent CB1 receptor agonist (Ki = 2.2 nM)that exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo. Learn MoreStarting at: $99.00
-
Bucindolol
Bucindolol is a non-selective β-adrenoceptor antagonist with additional α1-adrenoceptor blocking activity. Ki values are 1.61, 1.20 and 68.9 nM for β1-, β2- and α1-adrenoceptors respectively. Learn MoreStarting at: $139.00
-
GGTI 297
GGTI 297 is a geranylgeranyltransferase I (GGTase-I) inhibitor (IC50 values are 135 and 418 nM for GGTase-I and FTase inhibition respectively), which inhibits RhoA prenylation leading to inactivation of RhoA/ROCK and a decrease in basal tone of the internal anal sphincter in vitro. Learn MoreStarting at: $149.00
-
Noladin ether
Noladin ether is an endogenous agonist for the GPR55 and CB1 receptors (EC50 values are 10 and 37 nM respectively) that displays selectivity over CB2 receptors (Ki values are 21.2 nM and > 3mM at CB1 and CB2 respectively). Learn MoreStarting at: $98.00
-
Pronethalol hydrochloride
Pronethalol hydrochloride is a ??-adrenergic antagonist, clinically effective in the treatment of angina pectoris and some arrhythmias. Learn MoreStarting at: $69.00
-
N-Benzylnaltrindole hydrochloride
N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist with a long duration of action in vivo. Learn MoreStarting at: $95.00
-
(RS)-PPG
(RS)-PPG is a potent and selective group III metabotropic glutamate receptor agonist, with approximately 25-fold preference for hmGlu8. Learn MoreStarting at: $100.00
-
Dihydrexidine hydrochloride
Dihydrexidine hydrochloride is a potent, full efficacy dopamine D1 agonist which shows no agonist activity at peripheral D2 receptors or adrenoceptors at doses which cause maximal stimulation of D1 sites. Learn MoreStarting at: $95.00
-
GR 79236
GR 79236 is a adenosine A1 receptor agonist (Ki = 3.1 nM). Learn MoreStarting at: $155.00
-
TCN 238
TCN 238 is a positive allosteric modulator of mGlu4 receptors (EC50 = 1.0 μM for human and rat mGlu4 receptors). Learn MoreStarting at: $105.00
-
NPEC-caged-(S)-3,4-DCPG
NPEC-caged-(S)-3,4-DCPG is a (S)-3,4-DCPG caged with the photosensitive 1-(2-nitrophenyl)ethoxycarbonyl group. Learn MoreStarting at: $215.00
-
VU 0155041 sodium salt
VU 0155041 sodium salt is a potent, positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50 = 798 and 693 nM at human and rat mGlu4 receptors respectively). Learn MoreStarting at: $50.00
-
SCH 23390 hydrochloride
SCH 23390 hydrochloride is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types respectively). Learn MoreStarting at: $90.00
-
Arvanil
Arvanil is a cannabinoid CB1 and vanilloid TRPV1 (VR1) agonist (Ki values are 0.5 and 0.3 μM respectively), which also inhibits the anandamide transporter (IC50 = 3.6 μM). Learn MoreStarting at: $50.00
-
BNTX maleate
BNTX maleate is a standard selective δ1 opioid receptor antagonist, which inhibits neurogenic ion transport mediated by a putative novel opioid receptor in porcine ileal mucosa. Learn MoreStarting at: $115.00
