7-TM Receptors
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SDM25N hydrochloride
SDM25N hydrochloride is a potent and highly selective non-peptide δ receptor antagonist (Ki values are 4.7, 3800 and 7900 nM for δ, κ and μ receptors respectively). Learn MoreStarting at: $125.00
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Propranolol hydrochloride
Propranolol hydrochloride is a β-adrenergic antagonist. Learn MoreStarting at: $59.00
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Propranolol glycol
Propranolol glycol is a metabolite of propranolol. Learn MoreStarting at: $99.00
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trans-Triprolidine hydrochloride
trans-Triprolidine hydrochloride is a potent H1 receptor antagonist. Learn MoreStarting at: $42.00
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McN-A 343
McN-A 343 is a selective muscarinic M1 receptor agonist with selectivity for M1 over other muscarinic receptor types appears to arise from a high efficacy at M1 receptors. Learn MoreStarting at: $37.00
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SKF 83959 hydrobromide
SKF 83959 hydrobromide is a dopamine D1-like receptor partial agonist that act as an antagonist in vivo, producing anti-Parkinsonian effects and antagonizing the behavioral effects of cocaine. Learn MoreStarting at: $139.00
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SKF 38393 hydrobromide
SKF 38393 hydrobromide is a prototypical D1-like dopamine receptor selective partial agonist. Learn MoreStarting at: $109.00
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PF 514273
PF 514273 is a potent and selective CB1 receptor antagonist that inhibits food intake in vivo following oral administration. Learn MoreStarting at: $139.00
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1,3-Dipropyl-8-phenylxanthine
1,3-Dipropyl-8-phenylxanthine is a selective A1 adenosine antagonist. Learn MoreStarting at: $95.00
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FIT
FIT is a selective and irreversible δ-opioid agonist that acts by alkylating the receptor. Learn MoreStarting at: $139.00
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MJ 15
MJ 15 is a potent and selective CB1 receptor antagonist that inhibits food intake and increases in body weight in diet-induced obese rats and mice. Learn MoreStarting at: $139.00
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AMN 082 dihydrochloride
AMN 082 dihydrochloride is the first selective mGlu7 agonist, which potently inhibits cAMP accumulation and stimulates GTPγS binding in recombinant cells and on membranes expressing mGlu7 (EC50 = 64 - 290 nM). Learn MoreStarting at: $89.00
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Nitrocaramiphen hydrochloride
Nitrocaramiphen hydrochloride is a muscarinic antagonist with 71-fold selectivity for M1 over M2. Learn MoreStarting at: $95.00
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SKF 83566 hydrobromide
SKF 83566 hydrobromide is a potent and selective D1-like dopamine receptor antagonist (Ki~ 0.56 nM for D1; KB = 2 μM for D2). Learn MoreStarting at: $79.00
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LY 379268 disodium salt
LY 379268 disodium salt is a sodium salt of LY 379268, a highly selective group II mGlu receptor agonist. Learn MoreStarting at: $295.00
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SKF 83822 hydrobromide
SKF 83822 hydrobromide is a high affinity, selective dopamine D1-like receptor agonist. Learn MoreStarting at: $139.00
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SKF 81297 hydrobromide
SKF 81297 hydrobromide is a dopamine D1-like receptor agonist. Learn MoreStarting at: $149.00
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Histamine dihydrochloride
Histamine dihydrochloride is an an endogenous agonist at histamine receptors (H1-4) that stimulates gastric acid secretion and acts as a neurotransmitter in vivo. Learn MoreStarting at: $41.00
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Mepyramine maleate
Mepyramine maleate is a selective inverse agonist for the H1 receptor that Inhibits histamine induced inositol phosphate (InsP) production (log EC50 = -7.94) and intracellular calcium mobilization. Learn MoreStarting at: $50.00
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Cinnabarinic acid
Cinnabarinic acid is a mGlu4 receptor agonist that activates mGlu4 receptors in transiently transfected HEK293 cells, decreases cAMP levels in native cultured cerebellar granule cells and also counteracts excitotoxic neuronal cell death induced by NMDA in mixed cultures of cortical cells. Learn MoreStarting at: $129.00