Urotensin-II Receptor
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SB 611812
SB 611812 is an urotensin-II (UT) antagonist, which inhibits urotensin-II-induced proliferation of neonatal cardiac fibroblasts. Learn MoreStarting at: $139.00
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SB 657510
SB 657510 is a selective urotensin-II (UT) receptor antagonist (Ki values are 61, 17, 30, 65 and 56 nM at human, monkey, cat, rat and mouse receptors respectively), which inhibits U-II-induced intracellular Ca2+ mobilization (IC50 = 180 nM) and antagonizes the contractile action of U-II in isolated mammalian arteries and aortae (EC50 = 50 - 189 nM). Learn MoreStarting at: $139.00
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(±)-AC 7954 hydrochloride
(±)-AC 7954 hydrochloride is a highly selective, non-peptide urotensin-II (UT) receptor agonist that displays potent activity at human and rat UT receptors (pEC50 values are 6.5 and 6.7 respectively). Learn MoreStarting at: $139.00
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SB 706375
SB 706375 is a high affinity, non-peptide antagonist of the urotensin-II (UT) receptor with high affinity for mammalian UT receptors, including human, mouse and rat (Ki values are 9.3, 19.1 and 20.7 nM respectively, in HEK293 cells expressing recombinant UT receptors). Learn MoreStarting at: $139.00