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Transporters
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OMDM-2
OMDM-2 is a metabolically stable inhibitor of anandamide cellular uptake that displays relatively low affinity for CB1 and CB2 receptors with Ki values of 5.1 and > 10 μM and for vanilloid VR1 receptors with EC50 value of 10 μM. Learn MoreStarting at: $65.00
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Benzamil
Talampanel is a non-competitive AMPA/kainate receptor antagonist that displays 2.3-3-fold more potent activity than GYKI 52466 . Learn MoreStarting at: $50.00
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O-2093
O-2093 is an inhibitor of anandamide uptake (IC50 = 17.3 μM) with little or no activity at CB1, CB2, TRPV1 and FAAH. Learn MoreStarting at: $99.00
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SN-6
SN-6 is a selective Na+/Ca2+-exchange (NCX) inhibitor which displays some selectivity for NCX1. IC50 values are 2.9, 16 and 8.6 μM for inhibition of intracellular Na+-dependent 45Ca2+ uptake by cells expressing NCX1, NCX2 and NCX3 respectively. Learn MoreStarting at: $115.00
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UCM 707
UCM 707 is a potent endocannabinoid transport inhibitor. IC50 values are 0.8 and 30 μM for inhibition of the anandamide transporter and FAAH respectively. Ki values are 4700, 67 and > 5000 nM for CB1, CB2 and VR1 receptors respectively. Learn MoreStarting at: $125.00
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VDM 11
VDM 11 is a potent and selective inhibitor of the anandamide membrane transporter (AMT) with IC50 values of 4-11 μM, which displays negligible agonist activity at the hVR1 receptor and very weak action at CB1 and CB2 receptors. Learn MoreStarting at: $75.00
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AM 1172
AM 1172 metabolically stable anandamide uptake inhibitor (IC50 = 2.1 - 2.5 μM) and fatty acid amide hydrolase (FAAH) inhibitor (Ki = 3.18 μM). Learn MoreStarting at: $139.00
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AM 404
AM 404 is a competitive and selective inhibitor of carrier-mediated anandamide transport (IC50 = 1 μM). Does not activate CB1 receptors or inhibit anandamide hydrolysis but has been shown to activate native and cloned vanilloid receptors (pEC50 = 7.4). Active in vivo. Also available in water soluble emulsion . Learn MoreStarting at: $65.00
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Bupropion hydrochloride
Bupropion hydrochloride is a non-selective inhibitor of dopamine and noradrenalin transporters (Ki values are 1.4, 2.8 and 45 μM for NET, DAT and SERT transporters respectively), which also inhibits neuronal nicotinic acetylcholine receptors. Learn MoreStarting at: $99.00
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Nomifensine
Nomifensine is a potent inhibitor of noradrenalin and dopamine uptake (Ki values are 4.7, 26 and 4000 nM for inhibition of noradrenalin, dopamine and 5-HT uptake respectively, in rat brain), which increases central dopamine levels in rats following systemic administration. Learn MoreStarting at: $79.00
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Cocaine hydrochloride
Cocaine hydrochloride, a competitive inhibitor of monoamine neurotransmitter transporters, inhibits dopamine (DAT), serotonin (SERT) and noradrenalin (NET) transporters with Ki values are 267, 392 and 872 nM respectively. Learn MoreStarting at: $79.00
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GBR 12783 dihydrochloride
GBR 12783 dihydrochloride is a potent and selective inhibitor of dopamine uptake with IC50 value of 1.8 nM for inhibition of [3H]-dopamine uptake in rat striatal synaptosomes. Learn MoreStarting at: $99.00
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GBR 13069 dihydrochloride
GBR 13069 dihydrochloride is a potent inhibitor of dopamine uptake with an IC50 value of 40 nM. Learn MoreStarting at: $89.00
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Threo-methylphenidate hydrochloride
Psychomotor stimulant. Inhibitor of dopamine and noradrenalin transporters that increases the extracellular concentration of dopamine and noradrenalin. Learn MoreStarting at: $85.00
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Zoniporide dihydrochloride
Zoniporide dihydrochloride is a sodium-hydrogen exchanger isoform 1 (NHE1) inhibitor that displays selectivity over other NHE isoforms (Ki values are 14, 2200 and 220000 nM for human NHE1, human NHE2 and rat NHE3 respectively). Learn MoreStarting at: $140.00
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BTCP maleate
BTCP maleate is a potent dopamine re-uptake inhibitor with a behavioral profile different from that of PCP and similar to that of cocaine. Learn MoreStarting at: $95.00
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Mephedrone hydrochloride
Mephedrone hydrochloride Inhibits striatal dopamine uptake and hippocampal 5-HT uptake in synaptosomes (IC50 values are 467 and 558 nM respectively). Learn MoreStarting at: $95.00
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3-CPMT
3-CPMT binds with high affinity to the dopamine transporter (Ki = 30 nM) and blocks re-uptake of dopamine. Learn MoreStarting at: $50.00
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JHW 007 hydrochloride
JHW 007 hydrochloride is a dopamine uptake inhibitor which displays high affinity for the dopamine transporter (DAT) (Ki = 25 nM compared to 1330 and 1730 for NET and SERT respectively), and suppresses the effects of cocaine administration in a dose-dependent manner. Learn MoreStarting at: $120.00
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3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride
3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride is a potent inhibitor of dopamine uptake and transport (Ki = 11.8 nM). Learn MoreStarting at: $75.00
