Retinoid X Receptors

9 Item(s)

per page

  • Fluorobexarotene

    Fluorobexarotene is a RXR agonist (Ki = 12 nM; EC50 = 43 nM at RXRα receptors), which displays similar RAR agonist activity to bexarotene; exhibits an apparent RXR binding affinity 75% greater than bexarotene. Learn More

    Starting at: $160.00

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  • SR 11237

    SR 11237 is a pan retinoid X receptor (RXR) agonist that is devoid of any RAR activity. Learn More

    Starting at: $135.00

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  • LG 100754

    LG 100754 is a novel RXR:PPARγ agonist; sensitizes PPARγ by enhancing its ligand binding activity which displays selectivity over other permissive heterodimers such as RXR:LXRα and RXR:BAR/FXR. Learn More

    Starting at: $140.00

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  • HX 531

    HX 531 is a potent RXR antagonist (IC50 = 18 nM). Learn More

    Starting at: $149.00

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  • HX 630

    HX 630 is a RXR agonist, which acts as a retinoid synergist and enhances the potency of AM 80 in a HL-60 cell differentiation assay. Learn More

    Starting at: $149.00

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  • CD 3254

    CD 3254 is a selective RXRα agonist; exhibits no activity at RARα, RARβ or RARγ receptors. Learn More

    Starting at: $135.00

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  • LG 101506

    LG 101506 is a selective RXR modulator (Ki values are 3, 9 and 11 for RXRα, RXRβ and RXRγ respectively), which displays poor binding affinity for RAR isoforms (Ki values are 2746, 3516 and >10,000 nM for RARα, RARβ and RARγ respectively). Learn More

    Starting at: $139.00

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  • Docosahexaenoic acid

    Docosahexaenoic acid is a endogenous omega-3 fatty acid. It acts as a selective retinoid X receptor (RXR) agonist that displays no activity at RAR, thyroid hormone receptor or the vitamin D receptor (VDR). Learn More

    Starting at: $75.00

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  • UVI 3003

    UVI 3003 is a RXR antagonist that displays high RXR binding affinity. Learn More

    Starting at: $115.00

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9 Item(s)

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