Prostanoid Receptors

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  • L-655,240

    L-655,240 is a potent and selective thromboxane A2/prostaglandin endoperoxide receptor antagonist. pA2 values are 8 - 8.4 in guinea pig smooth muscle; IC50 = 7 nM for inhibition of human platelet aggregation. Orally active in vivo. Learn More

    Starting at: $105.00

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  • Prostaglandin F2α

    Prostaglandin E2 and F2α receptor agonist. Naturally-occurring prostaglandin and potent vasoconstrictor. Learn More

    Starting at: $159.00

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  • 16,16-Dimethyl Prostaglandin E2

    16,16-Dimethyl Prostaglandin E2 is a synthetic derivative of prostaglandin E2, which increases embryonic stem cell (ESC) hematopoietic colony formation in mouse bone marrow. Learn More

    Starting at: $85.00

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  • GW 627368

    GW 627368 is a selective prostanoid EP4 receptor competitive antagonist with additional affinity at TP receptors (pKi values are 7.0 and 6.8 in competition radioligand bioassays). Learn More

    Starting at: $179.00

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  • (+)-Fluprostenol

    (+)-Fluprostenol, a prostaglandin F2α (FP) receptor agonist, stimulates intracellular calcium mobilization in cloned human ocular FP receptors, rat A7r5 cells and mouse 3T3 cells (EC50 values are 17.5, 19.1 and 37.3 nM respectively). Learn More

    Starting at: $55.00

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  • U 46619

    U 46619 is a stable synthetic analog of the endoperoxide prostaglandin PGH2 first prepared in 1975, and acts as a thromboxane A2 (TP) receptor agonist. Learn More

    Starting at: $109.00

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  • Misoprostol

    Misoprostol is a cytoprotective prostaglandin E1 analog with Ki values of 120, 250, 67 and 67 nM at cloned mouse EP1, EP2, EP3 and EP4 receptors respectively. Learn More

    Starting at: $99.00

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  • Sulprostone

    Sulprostone is a selective EP3 and EP1 receptor agonist and also is synthetic PGE2 analog and allodynic agent. Learn More

    Starting at: $119.00

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  • Epoprostenol

    Epoprostenol is a endogenous prostanoid that is a potent agonist at IP prostanoid receptors. Learn More

    Starting at: $389.00

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  • Ozagrel hydrochloride

    Ozagrel hydrochloride is a potent and selective inhibitor of thromboxane (TXA2) synthetase that inhibits platelet aggregation in vitro and arachidonate-induced arterial contraction in vivo. Learn More

    Starting at: $85.00

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  • TCS 2510

    TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM), which displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM. Learn More

    Starting at: $139.00

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  • L-798,106

    L-798,106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2 respectively). Learn More

    Starting at: $140.00

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  • SC 19220

    SC 19220 is a selective EP1 receptor antagonist (IC50 = 6.7 μM for inhibition of [3H]-PGE2 binding to EP1 transfected COS cells). Learn More

    Starting at: $129.00

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  • ICI 185,282

    ICI 185,282 is a potent thromboxane receptor antagonist. Learn More

    Starting at: $95.00

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  • AA 2414

    AA 2414 is a thromboxane A2 (TP) receptor antagonist, which inhibits platelet aggregation and bronchoconstriction induced by a TXA2 mimetic in guinea pigs. Learn More

    Starting at: $90.00

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  • ICI 192,605

    ICI 192,605 is a potent thromboxane A2 receptor (TP receptor) antagonist. Competitively inhibits contractile responses to U 46619. Learn More

    Starting at: $95.00

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  • L-670,596

    L-670,596 is a potent and selective thromboxane A2/prostaglandin endoperoxide receptor antagonist (IC50 = 5.5 nM), which inhibits U-44069-induced contractions of guinea pig trachea (pA2 = 9.0) and human platelet aggregation in vitro (IC50 = 6.5 nM). Learn More

    Starting at: $135.00

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  • Latanoprost

    Latanoprost is a FP prostaglandin receptor agonist, which exhibits agonist activity at EP1 and EP3 receptors and displays greater selectivity than prostanglandin F2α . Learn More

    Starting at: $175.00

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  • SC 51322

    SC 51322 is a potent EP1 prostanoid receptor antagonist (Ki = 13.8 nM), which displays analgesic properties in vivo. Learn More

    Starting at: $105.00

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  • SC 51089

    SC 51089 is a selective EP1 prostanoid receptor antagonist (Ki values are 1.3, 11.2, 17.5, 61.1, > 100, > 100, > 100, >100 and > 100 μM for EP1, TP, EP3, EP2, EP4, FP and DP receptors respectively). Learn More

    Starting at: $115.00

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