PPARγ

Pioglitazone hydrochloride

Pioglitazone hydrochloride is a selective PPARγ agonist (EC50 = 0.69 μM). Learn More

Starting at: $45.00

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nTZDpa

nTZDpa is a potent, selective non-thiazolidinedione PPARγ partial agonist (EC50 = 57 nM); produces ~25% maximum efficacy. Learn More

Starting at: $100.00

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GW 1929 hydrochloride

GW 1929 hydrochloride is a highly selective orally active peroxisome proliferator-activated receptor (PPAR)γ agonist (pEC50 values are 8.05, < 4 and < 4 for human PPARγ, PPARα and PPARδ receptors respectively). Learn More

Starting at: $135.00

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S26948

S26948 is a selective PPARγ agonist (EC50 = 8.83 nM), which drives normal adipocyte differentiation and exhibits a lipid-lowering effect; reduces atherosclerosis in E2-KI mice, and displays antidiabetic properties and improves hepatic insulin sensitivity in intralipid-infusion (IL) rats. Learn More

Starting at: $139.00

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BADGE

RS 39604 hydrochloride is a potent and selective 5-HT4 antagonist, with a pKi of 9.1 at 5-HT4 receptors in guinea pig striatal membranes and greater than 1000-fold selectivity over 5-HT1A, 2C, 3 and D1, D2, M1, M2, AT1, B1 and α1C receptors. Learn More

Starting at: $80.00

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Ciglitazone

Ciglitazone is a selective agonist at PPAR&gamma with an EC50 value of 3 μM in vivo. Learn More

Starting at: $139.00

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SR 202

SR 202 is a selective PPARγ antagonist that inhibits PPARγ-dependent adipocyte differentiation and growth in vitro and in vivo. Learn More

Starting at: $90.00

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