Orphan 7-TM Receptors
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3,5-DHBA
3,5-DHBA is a selective agonist of hydroxycarboxylic acid receptor 1 (HCA1, also known as GPR81) (EC50 ~150 μM), Inhibits lipolysis in wild-type mouse adipocytes. Learn MoreStarting at: $59.00
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TUG 891
TUG 891 is a potent GPR120 agonist (pEC50 values are 7.36 and 7.77 for human and mouse GPR120 respectively). Learn MoreStarting at: $120.00
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TC-O 9311
TC-O 9311 is a potent GPR139 agonist (EC50 = 39 nM in CHO-K1 cells expressing human GPR139), which displays no activity against a range of 90 diverse targets. Learn MoreStarting at: $119.00
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Grifolic acid
Grifolic acid is a selective partial GPR120 agonist that induces ERK and [Ca2+]i responses in cells expressing GPR120. Learn MoreStarting at: $119.00
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PF9 tetrasodium salt
PF9 tetrasodium salt is a potent agonist of GPR17 with an EC50 value of 36 pM. Learn MoreStarting at: $195.00