Non-selective Adenosine
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Caffeine
Caffeine is a central nervous system stimulant, which mobilizes calcium from intracellular stores and inhibits benzodiazepine binding to GABA receptors. Learn MoreStarting at: $69.00
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2-Chloroadenosine
2-Chloroadenosine is a metabolically stable analog of adenosine that behaves as an adenosine receptor agonist (Ki values are 300, 80 and 1900 nM for A1, A2A and A3 receptors respectively). Learn MoreStarting at: $75.00
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CGH 2466 dihydrochloride
Adenosine A1, A2B and A3 receptor antagonist (IC50 values are 19, 21, and 80 nM respectively). Also inhibits p38 MAPK (IC50 = 187 - 400 nM) and phosphodiesterase type 4D (IC50 = 22 nM). Learn MoreStarting at: $99.00
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NECA
NECA is a potent adenosine receptor agonist (Ki values are 14, 20 and 6.2 nM for human A1, A2A and A3 receptors respectively; EC50 = 2.4 μM for human A2B), which inhibits platelet aggregation and is centrally active in vivo. Learn MoreStarting at: $49.00
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XCC
XCC is an adenosine receptor antagonist (Ki values are 42, 68 and 1130 nM for A1, A2B and A2A receptors). Learn MoreStarting at: $95.00
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XAC
XAC is an adenosine receptor antagonist (IC50 values are 1.8 and 114 nM at A1 and A2 receptors respectively). Learn MoreStarting at: $95.00