Non-selective 5-HT2

Cinanserin hydrochloride

Cinanserin hydrochloride is a 5-HT2 antagonist. Learn More

Starting at: $90.00

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Metergoline

Metergoline is an antagonist at 5-HT1/5-HT2 with activity at 5-HT1D. Has moderate affinity for 5-HT6 and high affinity for 5-HT7. Learn More

Starting at: $50.00

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Org 37684

Org 37684 is an agonist of 5-HT2 receptors, which exhibits a rank order of potency of 5-HT2C >5-HT2B >5-HT2A (pEC50 values are 8.17, 7.96 and 7.11 respectively, in transfected CHO-K1 cells). Learn More

Starting at: $119.00

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DOB hydrochloride

DOB hydrochloride is a Selective 5-HT2 receptor agonist with Ki values of 0.44, 59, 69, 831 and 3700 nM for 5-HT2H, 5-HT2L, 5-HT2C, 5-HT1B and 5-HT1A receptors respectively. Learn More

Starting at: $99.00

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Amperozide hydrochloride

Amperozide hydrochloride is a typical antipsychotic that displays high affinity for 5-HT2 receptors and low affinity for D2 receptors. Learn More

Starting at: $99.00

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Mirtazapine

Mirtazapine is an antidepressant agent that enhances noradrenalin (NA) release in rat brain via inhibition of α2-adrenergic autoreceptors and displays only weak affinity for monoamine transporters. Learn More

Starting at: $85.00

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