You have no items in your shopping cart.
NMDA Receptors
-
Phencyclidine hydrochloride
Phencyclidine hydrochloride is a non-competitive NMDA receptor antagonist and sigma receptor agonist. Learn MoreStarting at: $55.00
-
cis-ACPD
cis-ACPD is a 1:1 mixture of (1R,3R)- and (1S,3S)-ACPD. Potent NMDA receptor agonist and selective group II mGluR agonist (EC50 values are 13, 50, >300 and >300 μM at mGluR2, mGluR4, mGluR1 and mGluR5 respectively). Exhibits proconvulsant activity in vivo. Learn MoreStarting at: $125.00
-
DQP 1105
DQP 1105 is a noncompetitive NMDA receptor antagonist; displays over 50-fold selectivity for GluN2D- and GluN2C-containing receptors over GluN2B-, GluK2-, GluA1- and GluN2A-containing receptors (IC50 values are 2.7, 8.5, 121, 153, 198 and 206 μM respectively). Learn MoreStarting at: $119.00
-
(±)-1-(1,2-Diphenylethyl)piperidine maleate
(±)-1-(1,2-Diphenylethyl)piperidine maleate is a high affinity antagonist at the ion channel on the NMDA receptor. Learn MoreStarting at: $85.00
-
Norketamine hydrochloride
Norketamine hydrochloride is a major metabolite of ketamine that is a potent non-competitive NMDA receptor antagonist (Ki = 3.6 μM for displacement of [3H]-MK 801 in rat brain). Learn MoreStarting at: $99.00
-
(S)-(+)-Ketamine hydrochloride
(S)-(+)-Ketamine hydrochloride is a NMDA receptor antagonist, which displays neuroprotective efficacy in vitro. Learn MoreStarting at: $85.00
-
Spermidine trihydrochloride
Spermidine trihydrochloride binds to the polyamine modulatory site of the NMDA receptor and has been described as an agonist based on its ability to enhance the binding of [3H]-MK801. Learn MoreStarting at: $65.00
-
D-Serine
D-Serine is a glycine agonist at the NMDA receptor. L-Serine also available. Learn MoreStarting at: $79.00
-
Spermine tetrahydrochloride
Spermine tetrahydrochloride is a polyamine which produces a variety of modulatory effects on the NMDA receptor channel, acting through a specific site on the complex which can cause both agonist and antagonist effects. Learn MoreStarting at: $59.00
-
TCS 46b
Orally active, subtype-selective NR1A/NR2B NMDA receptor antagonist (IC50 values are 5.3, 35000 and > 100000 nM for NR1A/2B, NR1A/2A and NR1A/2C receptor subtypes respectively), whih potentiates the effect of L-DOPA in 6-OHDA-lesioned rats following oral administration. Learn MoreStarting at: $109.00
-
Synthalin sulfate
Synthalin sulfate is an effective non-competitive NMDA receptor antagonist in vivo and in vitro. Learn MoreStarting at: $85.00
-
Ifenprodil hemitartrate
Ifenprodil hemitartrate is a NMDA receptor antagonist, acting at the polyamine site. Learn MoreStarting at: $65.00
-
ACBC
ACBC is a NMDA receptor partial agonist, acting at the glycine site of NR1. Learn MoreStarting at: $80.00
-
CGP 78608 hydrochloride
CGP 78608 hydrochloride is a potent and selective NMDA antagonist that acts through the glycine site (IC50 = 5 nM). Displays > 500-fold selectivity over kainate and AMPA receptors (IC50 values are 2.7 and 3 μM respectively). Learn MoreStarting at: $140.00
-
Ro 8-4304 hydrochloride
Ro 8-4304 hydrochloride is a NMDA receptor antagonist (IC50 = 0.4 μM) that displays > 100 fold selectivity for NR2B-containing receptors over NR2A-containing receptors, which exhibits an activity-dependent mechanism of NMDA antagonism and is competitive with respect to spermine. Learn MoreStarting at: $109.00
-
Ro 04-5595 hydrochloride
Ro 04-5595 hydrochloride is a selective antagonist for NR2B-containing NMDA receptors (Ki = 31 nM). Learn MoreStarting at: $129.00
-
CIQ
CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit, which increases channel opening efficiency and enhances NMDA receptor responses. Learn MoreStarting at: $119.00
-
Homoquinolinic acid
Homoquinolinic acid is a potent NMDA receptor agonist; subtype-selective. Learn MoreStarting at: $129.00
-
Quinolinic acid
Quinolinic acid is an endogenous NMDA agonist and transmitter candidate. Learn MoreStarting at: $59.00
-
MNI-caged-D-aspartate
MNI-caged-D-aspartate is a D-aspartate caged with the photosensitive 4-methoxy-7-nitroindolinyl group. Learn MoreStarting at: $149.00
